Results 121 to 130 of about 2,283,209 (217)

SOM3355: a unique pharmacological profile combining VMAT1 inhibition, VMAT2-mediated dopamine modulation, and β₁-adrenergic antagonism for the treatment of movement and neuropsychiatric disorders. [PDF]

Front Pharmacol
Turilli-Ghisolfi ES, Støve SI, Huertas O, Kråkenes TA, Teigen K, Panigone S, Medori R.   +6 more
europepmc   +1 more source

Development of Novel Pegylated Imidazobenzodiazepines Targeting α5 GABAA Receptors for Anxiety: A Comparative Prodrug and Metabolite Study. [PDF]

ACS Chem Neurosci
Toriola MA, Kowalczyk ET, Medubi KM, Meyer MJ, Fernando MRT, Scholze P, Premananda N, Harrington SG, Barkley BR, Webb DA, Arnold LA.   +10 more
europepmc   +1 more source

The Selectivity Implications of Docking Libraries with Greater and Lesser Similarities to Bio-like Molecules. [PDF]

J Med Chem
Hall BW, Sakamoto K, Huang XP, Irwin JJ, Shoichet BK, Roth BL.   +5 more
europepmc   +1 more source

Thyroxin displacement from single and combined thyroid hormone binding proteins by various test substances. [PDF]

Arch Toxicol
Brandt J, Fabian E, Aktalay-Hippchen A, Jedermann L, Landsiedel R.   +4 more
europepmc   +1 more source

The Emergence of Isotryptamine Analogs as Novel Serotonergic Agents with Psychotherapeutic Potential. [PDF]

ACS Pharmacol Transl Sci
Glennon RA, Dukat M.
europepmc   +1 more source

A new radioligand binding assay to measure the concentration of drugs in rodent brain ex vivo. [PDF]

J Pharmacol Exp Ther, 2012
Hussmann GP, Kellar KJ.
europepmc   +1 more source

AB-MDMSBA-Not a Synthetic Cannabinoid Receptor Agonist. [PDF]

Pharmacol Res Perspect
Patel M, Ganeshan D, Horgan I, Partington H, Glass M.   +4 more
europepmc   +1 more source

A Structure-Activity Relationship Study of Alpha Synuclein PET Radiotracer M503-1619. [PDF]

Molecules
Tian GL, Hsieh CJ, Saturnino Guarino D, Lengyel-Zhand Z, Chia WK, Li S, Graham TJA, Hou C, Lee H, Young AJ, Petersson EJ, Mach RH.   +11 more
europepmc   +1 more source

Automated Parallel Synthesis Accelerates Virtual Screening Hit Discovery. [PDF]

J Am Chem Soc
McKenna SM, Šícho M, van der Horst C, Maasland J, van der Nol E, Turco G, Bernatavicius A, van Westen GJP, Heitman LH, Pomplun SJ.   +9 more
europepmc   +1 more source

Development and Biological Characterization of Fluorescent Dynorphins for the Visualization of Kappa Opioid Receptors. [PDF]

J Med Chem
Kalaba P, Böhm MP, D̵ikić F, Tomašević N, Drdla-Schutting R, Hasinger S, Ines DM, Wolf A, Belil-Catalina M, Bryant SD, Spetea M, Gruber CW, Muttenthaler M, Keimpema E.   +13 more
europepmc   +1 more source