Results 91 to 100 of about 4,042 (165)

Carbonic anhydrase inhibitors: Aliphatic N-phosphorylated sulfamates - A novel zinc-anchoring group leading to nanomolar inhibitors

, 2004
A small library of phosphorylated sulfamates (N-(O-alkylsulfamoyl)-phosphoramidic acids) incorporating long aliphatic chains (C8-C16) has been synthesized and investigated for their interaction with two physiologically relevant carbonic anhydrase (CA ...
Barragan, V, Supuran, CT, Montero, Jean-Louis, Bonnac, L, Innocenti, A, Bonnac, Laurent, Scozzafava, Andrea, Supuran, Claudiu,, Montero, JL, Innocenti, Alessio, Winum, JY, Casini, Angela, Barragan, Véronique, Scozzafava, A, Winum, Jean-Yves   +14 more
core   +1 more source

Synthesis and Applications of Sulfamates and Related Functionalities

Sulfur-containing moieties play a crucial role in both medicinal and synthetic chemistry. Chapters 2 and 3 focus on two sulfonamide bioisosteres called sulfamates and sulfamides.
Sguazzin, Matthew
core   +1 more source

Intramolecular PhIO Mediated Copper-Catalyzed Aziridination of Unsaturated Sulfamates: A New Direct Access to Polysubstituted Amines from Simple Homoallylic Alcohols

, 2016
Olefinic sulfamates derived from primary and secondary alcohols undergo intramolecular copper-catalyzed aziridination in the presence of iodosylbenzene to afford novel bicyclic fused aziridines.
Alberto Ghini (3065124), Robert H. Dodd (255173), Gerardo Burton (240155), Fernando Duran (3065118), Philippe Dauban (255170), Loïc Leman (3065121)   +5 more
core   +1 more source

A Multifunctional Sulfur(VI) Fluoride for SuFEx Reactions: N-CF₂H Sulfamoyl Fluorides. [PDF]

Angew Chem Int Ed Engl
Long Y, He X, Zhong W, Nie H, Deng L, Tao M, Lai Y, Sun C, Qian J, Zha Z, Zhang X, Liu J.   +11 more
europepmc   +1 more source

C(sp²)-C(sp²) and C(sp²)-C(sp³) Nickel-Catalyzed Kumada-Corriu and Buchwald-Hartwig Cross-Coupling of Aryl Sulfamates Enabled by Sterically-Demanding, Electron-Rich IPr*^OMe N-Heterocyclic Carbenes. [PDF]

Catal Sci Technol
Kardela M, Szostak M, Bisz E.
europepmc   +1 more source

Efficient Synthesis of Novel Propargyl Sulfamate Derivatives and Their Potent Inhibitory Effects on Human Carbonic Anhydrase Isoenzymes. [PDF]

ACS Omega
Atmaca U, Bayrak S, Bayrak C.
europepmc   +1 more source

Steroidal A/B-ring fusion as a strategy for isoform-selective inhibition of human carbonic anhydrases. [PDF]

RSC Adv
Brynda J, Kiss A, Pospíšilová K, Kapras V, Sieglová I, Slavíková B, Řezáčová P, Kudová E.   +7 more
europepmc   +1 more source

Comparison of Alkyl-Bridged Bis(N-Heterocyclic Carbene) Nickel Precatalysts: Structure and Catalytic Activity in the Reductive Cleavage and Suzuki-Miyaura Reactions. [PDF]

ACS Omega
Zhang CS, Beams EC, Moffett AL, Luo C, McMillen CD, Chianese AR, Green KA.   +6 more
europepmc   +1 more source

Chemo- and enantioselective intramolecular silver-catalyzed aziridinations of carbamimidates. [PDF]

Chem Commun (Camb), 2023
Trinh TA, Fu Y, Hu DB, Zappia SA, Guzei IA, Liu P, Schomaker JM.   +6 more
europepmc   +1 more source

Skeletal Rearrangement of Biaryls via Rhodium-Azirine Intermediate: A Route to Solid-State Emissive Polycyclic Sulfamates. [PDF]

ACS Catal
Insa-Carreras N, Díaz-Jiménez À, Pinto A, Rodríguez L, Poater A, Roglans A, Pla-Quintana A.   +6 more
europepmc   +1 more source