Results 81 to 90 of about 4,042 (165)
Efficacious N-protection of O-aryl sulfamates with 2,4-dimethoxybenzyl groups
, 2012 Sulfamates are important functional groups in certain areas of current medicinal chemistry and drug development. Alcohols and phenols are generally converted into the corresponding primary sulfamates (ROSO2NH2 and ArOSO2NH2, respectively) by reaction ...
Annalisa Bertoli (16199546) +4 more
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Betulinyl Sulfamates as Anticancer Agents and Radiosensitizers in Human Breast Cancer Cells
, 2015 Betulinic acid (BA), a natural compound of birch bark, is cytotoxic for many tumors. Recently, a betulinyl sulfamate was described that inhibits carbonic anhydrases (CA), such as CAIX, an attractive target for tumor-selective therapy strategies in ...
Daniel Emmerich +7 more
core +1 more source
A Study of Aldehyde Derivatives of Metallic Sulfamates [PDF]
, 1949 Sulfamic acid at one time had no particular value, and very little was known about the physical and chemical properties of this acid. At the present time , however, this acid is a commercial product of considerable importance and extensive investigation ...
Morin, Edmond A.
core +1 more source
Palladium- and Nickel-Catalyzed Aminations of Aryl Imidazolylsulfonates and Sulfamates
, 2011 A nickel complex derived from dppf, along with NaOt-Bu as the base, allowed for challenging aminations of aryl sulfamates. An improved functional group tolerance is observed in novel palladium-catalyzed aminations of imidazolylsulfonates with rac-BINAP ...
Song, Weifeng +5 more
core +1 more source
, 2016 High-speed and scalable nickel-catalyzed cross-coupling of arylboronic acids with aryl carbamates and sulfamates is achieved by using sealed-vessel microwave ...
Christian Pilger (2162587) +2 more
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The ring opening of aziridines by pendant sulfamates is a viable strategy for the rapid preparation of vicinal diamines. Our reaction is compatible with both disubstituted cis- and trans-aziridines; unsubstituted, N-alkyl, and N-aryl sulfamates engage ...
Someshwar Nagamalla (11965760) +4 more
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Palladium-Catalyzed Intramolecular Diamination of Acrylic Esters Using Sulfamates as Nitrogen Source
, 2016 An intramolecular diamination of acrylates is reported using sulfamates as nitrogen sources. This reaction proceeds under palladium(II) catalysis with copper bromide as oxidant and gives rise to anti-configured 2,3-diamino carboxylates as bicyclic ...
Kilian Muñiz (1393558) +3 more
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Stereochemical Models for Rh-Catalyzed Amination Reactions of Chiral Sulfamates
, 2016 Oxidative C−H amination of chiral sulfamate esters using achiral Rh-carboxylate catalysts, PhI(OAc)2, and MgO occurs in high yield and with good to excellent diastereocontrol. A number of examples are included to support a proposed transition state model
Jihee Lee (2432605) +2 more
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, 2016 Efficient bis(phosphine)nickel-catalyzed cross-couplings of diarylborinic acids with aryl chlorides, tosylates, and sulfamates have been effected with an assistance of N-heterocyclic carbene (NHC) generated in situ from N,N′-dialkylimidazoliums, e.g ...
Haihua Ke (1771690) +2 more
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, 2003 A series of aliphatic sulfamates and related derivatives incorporating cyclic/polycyclic (steroidal) moieties in their molecules has been synthesized and assayed as inhibitors of the zinc enzyme carbonic anhydrase (CA) and, more precisely, of the ...
Vullo, Daniela +10 more
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