Results 71 to 80 of about 13,320 (204)
, 2016 The hydrozirconation reaction of 1-alkynyl sulfoxides or sulfones with Cp2Zr(H)Cl in THF at room temperature predominantly gave Z-β-zirconated vinyl sulfoxides or sulfones with excellent regioselectivity.
Dehui Duan (2419603) +2 more
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A Facile and Mild Synthesis of Trisubstituted Allylic Sulfones from Morita-Baylis-Hillman Carbonates
Molecules, 2015 An efficient and catalyst-free synthesis of trisubstituted allylic sulfones through an allylic sulfonylation reaction of Morita-Baylis-Hillman (MBH) carbonates with sodium sulfinates has been developed.
Lin Jiang +5 more
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Multifunctional β-iodovinyl sulfones have emerged as versatile synthetic precursors, serving as key building blocks for diverse synthetic transformations.
Raghavaiah Pallepogu +3 more
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Dipolar addition to cyclic vinyl sulfones leading to dual conformation tricycles
Beilstein Journal of Organic Chemistry, 2013 Dipolar addition of cyclic azomethine imines with cyclic vinyl sulfones gave rise to functionalized tricycles that exhibited fluxional behavior in solution at room temperature.
Steven S. Y. Wong +4 more
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Synthesis of C2-symmetric bis-indolyl sulfones
, 2009 A new class of C2-symmetric bis-indole derivatives with 2,2-linkage has been synthesized from bis-propargyl sulfones. The method involves treatment of the sulfones with catalytic amount of triethylamine to form the indole derivatives presumably via the ...
Mitra, Tapobrata +5 more
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Spatial structure of α-halogen-substituted sulfones [PDF]
, 1981 1. Conformational equilibrium between the gauche- and trans-forms is attained in α-halogenated sulfones with the gauche-form predominating. 2. The position of the aryl radical in α-haloaryl sulfones is close to interfering with.
Vereshchagin A. +2 more
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Molecules, 2016 We reported herein the synthesis, antifungal activity, docking and in silico ADME prediction studies of four novel series of sulfones 6a–f, 8a–c, 10a–f and 12a–c.
Mohamed Fares +8 more
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Vinyl sulfones: selective and tunable covalent warheads against challenging enzyme targets [PDF]
Exploration of Drug ScienceOver the past several decades there has been a growing recognition of the role that covalent drug candidates have played in the drug development process. With this recognition, compounds that are capable of selectively and irreversibly inactivating their
Ronald E. Viola
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, 2016 A general and efficient method for the rhodium-catalyzed enantioselective catalytic conjugate addition of organoboronic acids to α,β-unsaturated sulfones is described.
Pablo Mauleón (2462224) +3 more
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Hydrohalogenation Reactions of 1,2-Allenic Sulfones. A Novel Synthesis of 2-Haloallylic Sulfones
, 2016 Hydrohalogenation Reactions of 1,2-Allenic Sulfones.
Shengming Ma (1312428), Qi Wei (198826)
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