Results 11 to 20 of about 12,154 (204)

Bilateral simultaneous acute angle closure caused by sulphonamide derivatives: A case series

open access: yesIndian Journal of Ophthalmology, 2010
The sulphonamide group of drugs is implicated in bilateral acute angle closure (AAC) due to an idiosyncratic response. We report a series of three cases with bilateral AAC caused by different sulphonamide derivatives, their presentation and management.
Senthil Sirisha   +3 more
doaj   +1 more source

Sulphonamide resistant commensal Neisseria with alterations in the dihydropteroate synthase can be isolated from carriers not exposed to sulphonamides [PDF]

open access: yesBMC Microbiology, 2002
Background Development of sulphonamide resistance in Neisseria meningitidis has been suggested to involve horizontal DNA-transfer from a commensal Neisseria species.
Swedberg Göte, Qvarnström Yvonne
doaj   +2 more sources

New sulphonamide pyrolidine carboxamide derivatives: Synthesis, molecular docking, antiplasmodial and antioxidant activities.

open access: yesPLoS ONE, 2021
Carboxamides bearing sulphonamide functionality have been shown to exhibit significant lethal effect on Plasmodium falciparum, the causative agent of human malaria.
Efeturi A Onoabedje   +3 more
doaj   +2 more sources

Metformin and its sulphonamide derivative simultaneously potentiateanti-cholinesterase activity of donepezil and inhibit beta-amyloid aggregation

open access: yesJournal of Enzyme Inhibition and Medicinal Chemistry, 2018
The aim of this study was to assess in vitro the effects of sulphenamide and sulphonamide derivatives of metformin on the activity of human acetylcholinesterase (AChE) and butyrylcholinesterase (BuChE), establish the type of inhibition, and assess the ...
Magdalena Markowicz-Piasecka   +2 more
doaj   +2 more sources

Sulphonamide Resistance in Neisseria meningitidis and Commensal Neisseria Species [Elektronisk resurs]

open access: yes, 2003
Extensive use of the sulphonamide drugs against the bacterium Neisseria meningitidis has resulted in drug resistance development. Sulphonamide resistance in N.
Qvarnström, Yvonne,   +2 more
core   +9 more sources

Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors

open access: yesJournal of Enzyme Inhibition and Medicinal Chemistry, 2018
A small collection of 26 structurally novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group, were synthesised and tested in enzyme inhibition assays against the tumour-associated hCA IX enzyme.
Özlen Güzel-Akdemir   +4 more
doaj   +2 more sources

Reasoned opinion on the review of the existing maximum residue levels (MRLs) for cyazofamid according to Article 12 of Regulation (EC) No 396/2005 [PDF]

open access: yesEFSA Journal, 2012
According to Article 12 of Regulation (EC) No 396/2005, the European Food Safety Authority (EFSA) has reviewed the Maximum Residue Levels (MRLs) currently established at European level for the pesticide cyazofamid.
European Food Safety Authority
doaj   +1 more source

Potent carbonic anhydrase I, II, IX and XII inhibition activity of novel primary benzenesulfonamides incorporating bis-ureido moieties

open access: yesJournal of Enzyme Inhibition and Medicinal Chemistry, 2023
A novel series of twelve aromatic bis-ureido-substituted benzenesulfonamides was synthesised by conjugation of aromatic aminobenzenesulfonamides with aromatic bis-isocyanates.
Tuba Tekeli   +5 more
doaj   +1 more source

Development of Praziquantel sulphonamide derivatives as antischistosomal drugs

open access: yesJournal of Enzyme Inhibition and Medicinal Chemistry, 2022
The almost empty armamentarium to treat schistosomiasis, a neglected parasitic disorder caused by trematode flatworms of the genus Schistosoma, except Praziquantel (PZQ), urged to find new alternatives to fight this infection.
Andrea Angeli   +6 more
doaj   +1 more source

Evidence of sulphonamide residues by rapid laboratory test [PDF]

open access: yesMljekarstvo, 2004
In addition to the significant role in the treatment of bacterial diseases, primarily mastitis, intestinal infections and pneumonia, sulphonamides are used as fodder additives.
Damir Kaša
doaj   +2 more sources

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