A reported potent and selective reversible MAGL inhibitor fails to reproduce its claimed potency in two established in vitro assays, even when the previously reported substrate is used, while eight related analogs are likewise inactive. The findings highlight substantial assay‐dependent behavior and the need for careful validation before such compounds
Juha R. Savinainen +3 more
wiley +1 more source
Synthetic Cannabinoid Use and Sports-Related Concussion Risk Among US Adolescents: Implications for School Health Screening and Prevention. [PDF]
Kalra S, Nagaraja N, Kalra D.
europepmc +1 more source
Identification and Structural Elucidation of a New Synthetic Cannabinoid, MDMB-5'Br-PINACA, in Seized Herbal Materials. [PDF]
de Godoi AB +6 more
europepmc +1 more source
Exploring the Role of Leukocyte Telomere Length and Human Telomerase Reverse Transcriptase MNS16A Variant in Cannabis or Synthetic Cannabinoid Use Disorder. [PDF]
Pehlivan S +5 more
europepmc +1 more source
Abuse Potential and Neurotoxic Effects of the Synthetic Cannabinoid 4F-ABUTINACA Self-Administration in Adult Male Rats. [PDF]
Shi B +10 more
europepmc +1 more source
Physicochemical Characterization and Metabolites Identification of the Synthetic Cannabinoid MDMB-5'Br-PINACA Using <i>In Silico</i> and <i>In Vitro</i> Approaches. [PDF]
Godoi AB +5 more
europepmc +1 more source
Synthetic Cannabinoid AB-FUBINACA Negatively Impacted the Male Fertility and Induced Testicular Toxicity. [PDF]
Alzu'bi A +7 more
europepmc +1 more source
Intranasal naloxone to treat suspected synthetic cannabinoid overdose: A case report and literature review. [PDF]
Dickinson J, Buckley T.
europepmc +1 more source
Entomological consequences and toxicological detection of synthetic cannabinoid receptor agonists (SCRAs) in necrophagous larvae (Diptera: Calliphoridae). [PDF]
Blavier CAK +6 more
europepmc +1 more source

