A new method for the synthesis of heterocyclic systems containing tetrazole and tetrahydroisoquinoline is developed via the performance of one-pot Ugi-azide and Heck cyclization reactions.
Jiawei Niu +6 more
doaj +1 more source
Asymmetric Synthesis of Tetrahydroisoquinoline Alkaloids Using Ellman's Chiral Auxiliary
Chiral t -butylsulfinamide has been successfully employed for the stereoselective synthesis of 1-benzyl tetrahydroisoquinoline alkaloids. This is the first report on the synthesis of chiral 1-benzyltetrahydroisoquinoline natural products using tert ...
Y. Vikram Reddy +5 more
doaj +1 more source
(S)-4-tert-Butyl-2-(1,2,3,4-tetrahydroisoquinolin-3-yl)-1,3-thiazole
In the title compound, C16H20N2S, a potential tetrahydroisoquinoline (TIQ) thiazole ligand, the N-containing six-membered ring of the TIQ unit adopts a half-chair conformation. There are four molecules in the asymmetric unit.
Sunayna Pawar +3 more
doaj +1 more source
Synthesis of Some Novel 11b-Substituted Pyrimido[6,1-a]-isoquinoline Derivatives
A series of novel 11b-substituted 1,6,7,11b-tetrahydropyrimido[6,1-a]- isoquinoline-2,4-diones and 4-thioxo-1,3,4,6,7,11b-hexahydropyrimido[6,1-a]isoquinolin-2- ones were synthesized, utilizing two alternative strategies for ring closure of ...
Atanas P. Venkov +2 more
doaj +1 more source
Heterogeneous Catalysts in Pictet-Spengler-Type Reactions
Several solid catalysts were evaluated as an alternative for 1,2,3,4-tetrahydroisoquinoline synthesis by means of the Pictet-Spengler reaction. The reaction catalysed by a mixed oxide (Mg and Al) led to the best yield and good regioselectivity; using an ...
Rodolfo Quevedo +2 more
doaj +1 more source
Organophotocatalytic synthesis of phosphoramidates
We describe the use of visible light in conjunction with an organic dye for the synthesis of phosphoramidates. Cross dehydrogenative coupling reactions between phosphites and amines are reported using organic dyes and light as catalysts for the first ...
Hao, Guo +5 more
core +1 more source
Selective N-alkylation of isoquinolines, benzazepines and thienopyridines with aromatic aldehydes and naphthols [PDF]
Fülöp, Ferenc +2 more
core +2 more sources
Antidepressant-Like Effect of the Endogenous Neuroprotective Amine, 1MeTIQ in Clonidine-Induced Depression: Behavioral and Neurochemical Studies in Rats [PDF]
Agnieszka Wąsik +3 more
core +1 more source
Chromophore content and molar absorptivity of phytochrome in the Pr-Form [PDF]
Brandlmeier, Thomas +2 more
core +1 more source
Pyropheophytin a accompanies pheophytin a in darkened light grown cells of Euglena [PDF]
Rüdiger, W. +4 more
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