Results 111 to 120 of about 4,593 (180)

Synthesis and antiproliferative studies of 5-aryl-2-(3-thienylamino)-1,3,4- thiadiazoles

, 2014
A series of 5-aryl-2-(3-thienylamino)-1,3,4-thiadiazoles 3a-m were synthesized in good yields in two steps starting from thiophen-3- isothiocyanates.
Gadais, Charlène, Kirsch, Gilbert, Revelant, Germain, Mathieu, Véronique, Hesse, Stéphanie   +4 more
core   +1 more source

The palladium-catalyzed cross-coupling reactions of 3-chloro-4-halogeno-1,2,5-thiadiazoles

, 2003
3,4-Dichloro- and 3-chloro-4-halogeno-1,2,5-thiadiazoles (halogeno-: bromo- and iodo-) are involved in Pd-catalyzed cross-coupling reactions under Stille and Suzuki conditions.
Alain Merschaert, Merschaert, A., Hugo J. Gorissen, Gorissen, HJ.   +3 more
core   +1 more source

Design, Synthesis, and Biological Evaluation of Amide Derivatives of Coumarin-1,2,4-Thiadiazoles as Anticancer Agents. [PDF]

Chem Biodivers
Lingala AK, Murahari KK, Eppakayala L, Manchal R.   +3 more
europepmc   +1 more source

Development of a Late-Stage Functionalization Strategy to Access Diverse 3,5-Disubstituted 1,2,4-Thiadiazoles. [PDF]

J Org Chem
Dobria A, Petros ZA, Mickel P, Aldrich LN.   +3 more
europepmc   +1 more source

Recent Advances in the Synthesis and Applications of 1,2,3/1,2,5-Thiadiazole- and Benzo[<i>c</i>][1,2,5/1,2,3]thiadiazole-Type Compounds. [PDF]

Molecules
Quiroga D, Rodríguez D, Coy-Barrera E.
europepmc   +1 more source

An Imidazo[2,1-b][1,3,4]thiadiazole Derivative Inhibits the Virulence Factor α-Hemolysin by Blocking the Pullout of Its Stem Domain. [PDF]

ChemMedChem
Korotkov VS, Lukat P, Di Lucrezia R, Shekhar A, Degenhart C, Diestel R, Bilitewski U, Dinkel K, Blankenfeldt W, Brönstrup M.   +9 more
europepmc   +1 more source

Synthesis and characterization of FeCuAlO₄ as a reusable heterogeneous acidic nanocatalyst for preparation of 2-amino-1,3,4-thiadiazole derivatives in water. [PDF]

Sci Rep
Nikoo A.
europepmc   +1 more source

Design, Synthesis, and Investigation of the Biological Activities of New Thiadiazole Derivatives With Anticancer Effects. [PDF]

Chem Biol Drug Des
Özkay Y, Bal E, Kurban B, Osmaniye D, Özkan BNS, Kaplancıklı ZA.   +5 more
europepmc   +1 more source

Synthesis and biological screening of some halogenated thiadiazoles and triazoles

, 2010
89-95 Acid hydrazide 1 is treated with aryl isothiocyanates to get corresponding thiosemicarbazides 2. Compounds 2 in acidic medium give thiadiazoles 3 and in basic medium give triazoles 4. These compounds are synthesized by conventional method and ultra
Saji, George, Narwade, S K, Randhavane, P V, Karale, B K   +3 more
core  

Utility of 3-(2-oxo-2H-chromen-3-yl)-1-phenyl-1H-pyrazole-4-carbaldehyde in the synthesis of novel 1,3,4-thiadiazoles or 1,3-thiazoles and study their cytotoxic activity. [PDF]

Sci Rep
Abdel-Aziem A, Abdelhamid AO.
europepmc   +1 more source