Results 291 to 300 of about 44,050 (359)

Identification of a novel antifungal backbone of naphthalimide thiazoles with synergistic potential for chemical and dynamic treatment.

Future Medicinal Chemistry, 2021
Aim: The high incidence and prevalence of fungal infections call for new antifungal drugs. This work was to develop naphthalimide thiazoles as potential antifungal agents.
Peng-Li Zhang, G. Lavanya, Yang Yu, Bo Fang, Cheng‐He Zhou   +4 more
semanticscholar   +1 more source

Single-Pot Preparation of 4-Amino-2-(het)aryl-5-Substituted Thiazoles Employing Functionalized Dithioesters as Thiocarbonyl Precursors.

Journal of Organic Chemistry, 2021
An effective, diversity oriented, one-pot reaction of 4-amino-2-(het)aryl/alkyl-5-functionalized thiazoles has been disclosed, utilizing aryl/heteroaryl/alkyl dithioesters as thiocarbonyl coupling partners in a modified Thorpe-Ziegler type cyclization ...
Anusha Avadhani, P. Iniyavan, Y. Kumar, H. Ila   +3 more
semanticscholar   +1 more source

Synthesis, in‐vitro and in‐silico study of novel thiazoles as potent antibacterial agents and MurB inhibitors

Archiv der Pharmazie, 2020
Efficient procedures are herein reported for the synthesis of novel hybrid thiazoles via a one‐pot three‐component protocol. The protocol involves the reaction of novel aldehyde, thiosemicarbazide and halogen‐containing reagents in solvent‐ and catalyst ...
S. Sanad, Ahmed A. M. Ahmed, Ahmed E. M. Mekky   +2 more
semanticscholar   +1 more source

An unexpected discovery toward novel membrane active sulfonyl thiazoles as potential MRSA DNA intercalators.

Future Medicinal Chemistry, 2020
Aim: With the increasing emergence of drug-resistant bacteria, the need for new antimicrobial agents has become extremely urgent. This work was to develop sulfonyl thiazoles as potential antibacterial agents.
Yuan-Yuan Hu, Juan Wang, Tiejun Li, Rammohan R. Yadav Bheemanaboina, M. Ansari, Yu Cheng, Cheng‐He Zhou   +6 more
semanticscholar   +1 more source

Direct Arylation of Thiazoles on Water [PDF]

Angewandte Chemie, 2007
AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable via the “References” option.
Turner, Gemma L., Morris, James A., Greaney, Michael F.   +2 more
openaire   +2 more sources

Thiazoles and Thiazolidinones as Antioxidants

Current Medicinal Chemistry, 2013
Antioxidants are of great interest because of their involvement in important biological and industrial processes. According to Halliwell antioxidants are substances that at low concentration significantly delay or prevent oxidation. Chemically, oxidation is a process in which a loss of electrons occurs.
Athina Geronikaki, Konstantinos Liaras, Eleni Pitta   +2 more
openaire   +3 more sources

Synthetic and Medicinal Perspective of Fused-Thiazoles as Anticancer Agents.

Anti-Cancer Agents in Medicinal Chemistry, 2020
Fused triazole had explored their apartment as one of the important class of heterocycles, extensively used by chemists due to their diverse pharmacological activities in both synthetic organic chemistry and systemic biological field.
S. Pawar, Kapil Kumar, M. Gupta, R. Rawal   +3 more
semanticscholar   +1 more source

ChemInform Abstract: The Thiazole Aldehyde Synthesis [PDF]

ChemInform, 1998
AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable via the “References” option.
openaire   +3 more sources

Thiazole‐Mediated Synthetic Methodology

ChemInform, 2004
AbstractFor Abstract see ChemInform Abstract in Full Text.
DONDONI, Alessandro, MARRA, Alberto
openaire   +4 more sources

Cu-Catalyzed Aerobic Oxidative Sulfuration/Annulation Approach to Thiazoles via Multiple Csp3-H Bond Cleavage.

Organic Letters, 2018
A novel and practical Cu-catalyzed aerobic oxidative synthesis of thiazoles was developed. This chemistry for the first time achieved thiazole construction from simple aldehydes, amines, and element sulfur through multiple Csp3-H bond cleavage processes.
Xiaoyang Wang, Xu Qiu, Jialiang Wei, Jianzhong Liu, Song Song, W. Wang, N. Jiao   +6 more
semanticscholar   +1 more source