Results 111 to 120 of about 1,080,434 (247)

Design, synthesis, in vitro, and in silico studies of 4-fluorocinnamaldehyde based thiosemicarbazones as urease inhibitors

Scientific Reports
Clinically significant problems such as kidney stones and stomach ulcers are linked to the activation of the urease enzyme. At low pH, this enzyme gives an ideal environment to Helicobacter pylori in the stomach which is the cause of gastric ulcers and ...
Muhammad Islam, Saeed Ullah, Ajmal Khan, Zahra Batool, Suraj N. Mali, Shailesh S. Gurav, Kholood A. Dahlous, Saikh Mohammad, Javid Hussain, Ahmed Al-Harrasi, Zahid Shafiq   +10 more
doaj   +1 more source

Smart mesoporous silica nanoparticles for precision cancer therapy: Tumor targeting and stimuli‐responsive controlled release

Smart Molecules, EarlyView.
Smart mesoporous silica nanoparticles integrate tunable pore structures, molecular gates, targeting ligands, and stimuli‐responsive components to achieve controlled drug release for precision cancer therapy. This review highlights design principles, therapeutic applications, and future directions in immunotherapy, biodegradability, biosafety, and ...
Majdi Al‐Amili, Lei Lei, Zhu Jin
wiley   +1 more source

Synthesis, Density Functional Theory (DFT), Urease Inhibition and Antimicrobial Activities of 5-Aryl Thiophenes Bearing Sulphonylacetamide Moieties

Molecules, 2015
A variety of novel 5-aryl thiophenes 4a–g containing sulphonylacetamide (sulfacetamide) groups were synthesized in appreciable yields via Pd[0] Suzuki cross coupling reactions.
Mnaza Noreen, Nasir Rasool, Yasmeen Gull, Muhammad Zubair, Tariq Mahmood, Khurshid Ayub, Faiz-ul-Hassan Nasim, Asma Yaqoob, Muhammad Zia-Ul-Haq, Vincenzo de Feo   +9 more
doaj   +1 more source

Exploring the Synthetic Chemistry of Phenyl-3-(5-aryl-2-furyl)- 2-propen-1-ones as Urease Inhibitors: Mechanistic Approach through Urease Inhibition, Molecular Docking and Structure-Activity Relationship. [PDF]

Biomedicines, 2023
Fatima M, Aslam S, Zafar AM, Irfan A, Khan MA, Ashraf M, Faisal S, Noreen S, Shazly GA, Shah BR, Bin Jardan YA.   +10 more
europepmc   +1 more source

Herbivore and mesocarnivore carcasses trigger divergent short‐term changes in soil properties

Journal of Animal Ecology, EarlyView.
Scavengers reshape nutrient cycles in soils under carrion. Compared to herbivore carcasses, smaller but longer‐lasting carnivore remains boost nutrient levels and microbial activity in dry soils. Abstract Animal corpses act as pulses of organic matter (OM) and serve a key zoogeochemical role by providing localized nutrient inputs to soils and thereby ...
Adrián Colino‐Barea, Fuensanta García‐Orenes, Zebensui Morales‐Reyes, Moisés Gonzálvez, Carlos Martínez‐Carrasco, Marcos Moleón, Daniel Redondo‐Gómez, Evan A. N. Marks, Minerva García‐Carmona, Victoria Arcenegui, José Carlos Huerta‐del‐Bosque, Adrián Orihuela‐Torres, Santiago Soliveres, Sofia Albolafio, Esther Sebastián‐González, José Antonio Sánchez‐Zapata   +15 more
wiley   +1 more source

Alpinetin: anti-human gastric cancer potential and urease inhibition activity in vitro. [PDF]

Arch Med Sci, 2023
Zhang H, Jiang Q, Gong G, Li M, Alotaibi SH.   +4 more
europepmc   +1 more source

Stable flies preferentially oviposit on sites offering conspecific eggs with egg‐derived bacterial semiochemicals

Insect Science, EarlyView.
Stable flies preferentially oviposit on sites offering conspecific eggs with egg‐derived airborne semiochemicals. Egg‐borne bacterial symbionts, and Serratia marcescens in particular, produce odorants which attract gravid female flies and elicit oviposition.
Emmanuel Hung, Anya Gould, Stephanie Zaborniak, Caelen Watson, Regine Gries, Sukhmani Kaur, Kyra Stephens, Augustus Negraeff, Ryan Lam, Alpha Hui, Pantea Zamani, Aryan Monfared, Gerhard Gries   +12 more
wiley   +1 more source

Urease

, 2017
Although the discovery of urease as the first enzyme for which nickel is essential for activity dates back to 1975, the rationale for Ni selection for the active site of this hydrolase has been only recently unraveled.
L. Mazzei, F. Musiani, S. Ciurli, MAZZEI, LUCA, MUSIANI, FRANCESCO, CIURLI, STEFANO LUCIANO   +5 more
core   +1 more source

Investigation of Newly Synthesized Bis-Acyl-Thiourea Derivatives of 4-Nitrobenzene-1,2-Diamine for Their DNA Binding, Urease Inhibition, and Anti-Brain-Tumor Activities. [PDF]

Molecules, 2023
Arshad N, Parveen U, Channar PA, Saeed A, Saeed WS, Perveen F, Javed A, Ismail H, Mir MI, Ahmed A, Azad B, Khan I.   +11 more
europepmc   +1 more source

First Report of Tenacibaculum maritimum Infection in Grouper (Epinephelus spp.) Aquaculture in Taiwan

Journal of Fish Diseases, EarlyView.
ABSTRACT Between April 2024 and 2025, six independent outbreaks of ulcerative skin disease occurred in cultured groupers (Epinephelus spp.) across southern Taiwan and Penghu County during winter‐to‐spring seasonal transitions at water temperatures ranging from 19°C to 24°C.
Shang‐Ting Wu, Chia‐Yu Hsieh
wiley   +1 more source