Advances in chemistry and biological activity of fluorinated 1,3,5-triazines
The substitution of hydrogen by fluorine as bioisosteric replacement has been practised widely in agricultural and medicinal chemistry. This has led to the discovery of many pesticides and therapeutically useful chemical entities.
W. Chui (23304466) +2 more
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C-Ribosyl imidazo[2,1-f][1,2,4]triazines and 3-[2-(3-carboxyphenyl)ethyl]-3,6,7,8-tetrahydroimidazo[4,5-d][1,3]diazepin-8-ols represent two classes of known AMP deaminase inhibitors.
Stephen D. Lindell (2268556) +2 more
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Synthesis of C-(β-D-glucosaminyl)-1,2,4-triazines
In my diploma thesis I studied the syntheses of C-glucosaminyl-1,2,4-triazines and 1,2,4-triazin-5(4H)-ones. For the preparation of the target heterocycles C-(2-deoxy-2-phthalimido-3,4,6-tri-O-acetyl-β-D-glucopyranosyl)formamidrazone was prepared first ...
Hashimov, Mahir
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Design, Synthesis, and Antimicrobial Evaluation of New Annelated Pyrimido[2,1-c][1,2,4]triazolo[3,4-f][1,2,4]triazines. [PDF]
El Azab IH, Elkanzi NAA.
europepmc +1 more source
A CONVENIENT AND GENERAL SYNTHESIS OF THIADIAZOLO [2,3-C] [1,2,4] TRIAZINES [PDF]
Condensation and cyclization of 5-hydroxy- 1,2,4- thiadiazol-2-yl hydrazine 1 with pyruvic acid, phenacyl bromide, propargyl bromide and ally1 bromide afforded compounds 2,5,7 3, 4 ,6 and 8 respectively, Reaction of 1 with epichforohydrine afforded 4 ...
doaj
Synthesis, biological activity and molecular modeling study of novel 1,2,4-triazolo[4,3-b][1,2,4,5]tetrazines and 1,2,4-triazolo[4,3-b][1,2,4]triazines. [PDF]
El-Reedy AAM, Soliman NK.
europepmc +1 more source
The 5,7-diamino[1,2,4]triazolo[1,5-a][1,3,5]triazines were synthesized by cyclocondensation of 3(5)-amino-1,2,4-triazoles with cyanoguanidine. The substituted 3(5)-amino-1,2,4-triazoles were prepared from corresponding hydrazides and S-methylisothiourea ...
W. Chui (23304466) +2 more
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Synthesis and crystal structures of 6- and 8-methyl-3-phenyl-benzo[<i>e</i>][1,2,4]triazines. [PDF]
Constantinides CP +4 more
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General Synthesis of 1-Aryl-6-azaisocytosines and Their Utilization for the Preparation of Related Condensed 1,2,4-Triazines. [PDF]
Zálešák F, Slouka J, Stýskala J.
europepmc +1 more source
Synthesis, Properties, and Biological Activity Evaluation of Some Novel Naphtho[2,1-e]pyrazolo[5,1-c][1,2,4]triazines. [PDF]
Burcă I +6 more
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