Results 11 to 20 of about 18,197,302 (162)
SYNTHESIS OF NEW ACTIVATED INDOLES; 3-(4’-BROMOPHENYL)-4,6-DIMETHOXY-2-METHYLINDOLE [PDF]
Indonesian Journal of Chemistry, 2010 3-(4'-Bromophenyl)-4,6-dimethoxy-2-methylindole has been synthesized from 4,6-dimethoxyaniline via the modified Bischler method. Reaction of 4,6-dimethoxyaniline with 2,4-dibromopropiophenone gave an aniline ketone in 85%, and then it was protected to ...
Tutik Dwi Wahyuningsih
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Biotransformation of Indole to 3-Methylindole by Lysinibacillus xylanilyticus Strain MA [PDF]
Journal of Chemistry, 2015 An indole-biotransforming strain MA was identified as Lysinibacillus xylanilyticus on the basis of the 16S rRNA gene sequencing. It transforms indole completely from the broth culture in the presence of an additional carbon source (i.e., sodium succinate)
Pankaj Kumar Arora +3 more
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Pharmaceuticals, 2015 Seven novel N-arylsulfonyl-3-(2-yl-ethanone)-6-methylindole derivatives 4a–f and 6 were readily synthesized and have been identified as inhibitors of human immunodeficiency virus type-1 (HIV-1) replication. Initial biological studies indicated that among
Zhiping Che +5 more
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Influence of 3-acetyl-5-hydroxy-2-methylindole on glioma cell proliferation and metabolism
Журнал Белорусского государственного университета: Химия, 2022 A 3-acetyl analogue of 5-hydroxyindole was synthesised and evaluated for its effects on rat C6 glioma cell functions. It was found that 3-acetyl-5-hydroxy-2-methylindole at 10 μmol/L led to a sharp reduction of mitochondrial membrane potential, induction
Jan U. Panada +8 more
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3-Aryl-2H-azirines as annulation reagents in the Ni(II)-catalyzed synthesis of 1H-benzo[4,5]thieno[3,2-b]pyrroles [PDF]
Beilstein Journal of Organic ChemistryA high-yielding method for the synthesis of 3-arylbenzo[4,5]thieno[3,2-b]pyrroles has been developed via pyrrole ring annulation to the aromatic benzo[b]thiophene system, using 3-arylazirines as a N‒C=C synthon.
Julia I. Pavlenko +5 more
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Antibiofilm and Antivirulence Properties of Indoles Against Serratia marcescens
Frontiers in Microbiology, 2020 Indole and its derivatives have been shown to interfere with the quorum sensing (QS) systems of a wide range of bacterial pathogens. While indole has been previously shown to inhibit QS in Serratia marcescens, the effects of various indole derivatives on
Sivasamy Sethupathy +4 more
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Spectrophotometric study of the protonation processes of some indole derivatives in sulfuric acid [PDF]
Journal of the Serbian Chemical Society, 1999 The protonation of 3-methylindole, D-tryptophan, 3-formylindole, 3-acetylindole and indolyl-2-carboxylic acid in sulfuric acid media was studied by UV spectro-scopy.
GORAN M. STOJKOVIC +1 more
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The role of 3-methylindole in the aetiology of fog fever in cattle [PDF]
, 1981 3-Methylindole (skatole) is a metabolite of L-tryptophan formed in the rumen of cattle. There is considerable evidence that 3-methylindole is the cause of fog fever (acute bovine pulmonary emphysema) in cattle.
Hanafy, Mohamed Samih Mahmoud
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Molecules, 2022 A new synthetic alternative to the synthesis of 3-methyl indoles and 3-methyl indoline-2-ols with an excellent atomic economy is presented in this study.
Frank Hochberger-Roa +6 more
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Indole analogues decreasing the virulence of Vibrio campbellii towards brine shrimp larvae
Microbial Biotechnology, 2022 Indole signalling has been proposed as a potential target for the development of novel virulence inhibitors to control bacterial infections. However, the major structural features of indole analogues that govern antivirulence activity remain unexplored ...
Shanshan Zhang, Qian Yang, Tom Defoirdt
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