Antimicrobial activity of 1, 3, 4-thiadiazole derivatives: a recent review [PDF]
Journal of Applied Pharmaceutical Research, 2018 A few five members’ aromatic systems having three hetero-atoms at symmetrical positions, for example, thiadiazoles have been considered broadly attributable to their intriguing pharmacological properties.
Alam, Faruk
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Action of 2-Amino-1, 3, 4-thiadiazole in Controlling Plant Diseases
Japanese Journal of Phytopathology, 1971 Properties of 2-amino-1, 3, 4-thiadiazole (ATDA) as rice bacterial leaf blight controlling agent were examined.This compound was effective against the disease as foliar application, and also as root application.As foliar spray, ATDA showed immediate therapeutic effect, and the duration of the effect was fairly short.When applied into paddy water, ATDA ...
Kunito YAKUSHIJI, Osamu WAKAE
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A Convenient route for the synthesis of antimicrobial 1, 3, 4- thiadiazole derivatives
Bibechana, 2012 Thiosemicarbazide of 6-chloro-2- aminobenzothiazole on cyclization with different aromatic carboxylic acids in Phosphorus oxychloride provided the corresponding 2-aryl-5-(6’-chloro-1’,3’-benzothiazole-2-yl-amino)-1,3,4-thiadiazoles 4a-j. The compounds
AD Mishra
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Synthesis and Antimicrobial Activity of Some 2-[(4-Substituted-Phenyl-3-Chloro-Azetidin-2-One)-5-(2'-Methylamino-4-Phenyl-1', 3'-Thiazolyl-]-1, 3,4-Thiadiazoles [PDF]
Journal of Sciences, Islamic Republic of Iran, 2009 A new 2-[(4-substituted-phenyl-3-chloroazetidin-2-one)-5-(2'-methylamino 4-phenyl-1', 3'-thiazolyl-]-1, 3, 4-thiadiazoles, 5(a-n) were synthesized from 2-substituted-benzylideneamino-5-[2'-methylamino-4'-phenyl-1',3'-thiazolyl]-1,3, 4-thiadiazole, 4(a-n)
S.D. Srivastava
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Studies on 1, 3, 4-Thiadiazole Derivatives. VIII
YAKUGAKU ZASSHI, 1953 Masaki Ohta, Hiroshi Oya, Akira Mifune
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Synthesis and anticancer activity of some novel 3-(1, 3, 4-thiadiazol-2-yl)-quinazolin-4-(3H)-ones [PDF]
Orbital: The Electronic Journal of Chemistry, 2010 Quinazolinone is a versatile lead molecule for designing potential bioactive agents. The compounds that have quinazolin-4-ones moiety are associated with interesting biological activities such as antifungal, antibacterial, antiviral, antitubercular and ...
Alex Joseph +6 more
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Synthesis and Biological Evaluation of Some Newer 1H-Benzo[b][1,5]diazepin-2(3H)-one Derivatives as Potential Anticonvulsant Agents [PDF]
Pharmaceutical Sciences, 2022 Background: Regardless of the availability of all novel and earlier treatments, seizure control is notoriously complicated. In the hopes of discovering the latest and ultimate therapy, medicinal chemists will keep on to hunt for new antiepileptic ...
Dinesh D Rishipathak +2 more
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Design of 1-(furan-2-yl)-N-(5-substituted phenyl-1, 3, 4-thiadiazol-2-yl) methanimine derivatives as Enoyl-ACP reductase inhibitors: Synthesis, molecular docking studies and antitubercular activity [PDF]
Bangladesh Journal of Pharmacology, 2013 A series of 5-phenylsubstiuted 1, 3, 4 thiadiazoles clubbed with furan moiety (Fa-Fe) by means of azomethine linkage have been synthesized. All the newly synthesized compounds were characterized by IR,1HNMR and Mass analyses.
Bijo Mathew +5 more
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Фармацевтичний журнал, 2021 One of the promising methods of creating antitumor drugs is the screening of potential antitumor agents among synthesized compounds. Nitrogen-based heterocycle analogues are an extremely important class of organic substances that are widely used in ...
I. І. Myrko +4 more
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