Results 111 to 120 of about 79,681,589 (222)

Existence of Brain 5‑HT1A–5-HT2A Isoreceptor Complexes with Antagonistic Allosteric Receptor–Receptor Interactions Regulating 5‑HT1A Receptor Recognition

ACS Omega, 2017
Dasiel O. Borroto-Escuela, Xiang Li, Alexander O. Tarakanov, David Savelli, Manuel Narváez, Kirill Shumilov, Yuniesky Andrade-Talavera, Antonio Jimenez-Beristain, Bartosz Pomierny, Zaida Díaz-Cabiale, Riccardo Cuppini, Patrizia Ambrogini, Maria Lindskog, Kjell Fuxe   +13 more
doaj   +1 more source

Synthesis by microwave irradiation and binding properties of novel 5-HT1A receptor ligands.

, 2001
The synthesis by microwave irradn. and the binding tests on the 5-HT1A, 5-HT2A and 5-HT2C receptors of new substituted piperazines in order to identify selective ligands for 5-HT1A subtype receptor are reported. Conventional heating and microwave irradn.
Gessi S, Cattabriga E, SEVERINO, BEATRICE, FIORINO, FERDINANDO, SANTAGADA, VINCENZO, CALIENDO, GIUSEPPE, Borea P. A, PERISSUTTI, ELISA   +7 more
core  

Novel Potent 5-HT1a Agonists Selective over alpha1-Adrenoceptor Subtypes

, 2016
The analogues 2-5 of the potent 5-HT1A receptor agonist and α1d-adrenoceptor (α1d-AR) antagonist 1 (1) were rationally designed and prepared to preliminarily evaluate whether electronic and/or lipophilic properties of substituents in the ortho position
Micioni Di Bonaventura, Maria Vittora, BONIFAZI, ALESSANDRO, GIORGIONI, Gianfabio, Vistoli, Giulio, PETRELLI, Riccardo, Mazzolari, Angelica, DEL BELLO, FABIO, PIERGENTILI, Alessandro, Newman, Amy H., Keck, Thomas M., Poggesi, Elena, CIFANI, Carlo, QUAGLIA, Wilma, GIANNELLA, Mario, Cilia, Antonio   +14 more
core   +1 more source

Effect of 5-HT1A Receptor Partial Agonists of the Azapirone Class as an Add-On Therapy on Psychopathology and Cognition in Schizophrenia: A Systematic Review and Meta-Analysis. [PDF]

Int J Neuropsychopharmacol, 2023
Yamada R, Wada A, Stickley A, Yokoi Y, Sumiyoshi T.   +4 more
europepmc   +1 more source

Serotonin (5-HT1A) receptor [PDF]

Science-Business eXchange, 2011
openaire   +1 more source

Curated Database and Preliminary AutoML QSAR Model for 5-HT1A Receptor. [PDF]

Pharmaceutics, 2021
Czub N, Pacławski A, Szlęk J, Mendyk A.   +3 more
europepmc   +1 more source

(2,2-Diphenyl-[1,3]oxathiolan-5-ylmethyl)-(3-phenyl-propyl)-amine: a Potent and Selective 5-HT1A Receptor Agonist

, 2009
Starting from compound 1, a previously reported a1D-adrenocep- tors antagonist, a new series of ligands acting at 5-HT1A serotonin receptor were identified through simple structure modifications.
SORBI C., BRASILI L., TAIT A., MARUCCI, Gabriella, DE STEFANI C., FRANCHINI S., CILIA A., GALLESI R., PRANDI A., BUCCIONI, Michela   +9 more
core   +1 more source

Brain 5-HT1A Receptor PET Binding, Cortisol Responses to Stress, and the Familial Transmission of Suicidal Behavior. [PDF]

Int J Neuropsychopharmacol, 2022
Melhem NM, Zhong Y, Miller JM, Zanderigo F, Ogden RT, Sublette ME, Newell M, Burke A, Keilp JG, Lesanpezeshki M, Bartlett E, Brent DA, Mann JJ.   +12 more
europepmc   +1 more source

Serotonin (5-HT1A) receptor [PDF]

Science-Business eXchange, 2010
openaire   +1 more source

A new approach to 'on-demand' treatment of lifelong premature ejaculation by treatment with a combination of a 5-HT_1A receptor antagonist and SSRI in rats. [PDF]

Front Neurosci, 2023
Olivier JDA, Janssen JA, Esquivel-Franco DC, de Prêtre S, Olivier B.   +4 more
europepmc   +1 more source