Results 21 to 30 of about 4,308 (256)

Design, Synthesis, and Antifungal Activity of Some Novel Phenylthiazole Derivatives Containing an Acylhydrazone Moiety

Molecules, 2023
Crop fungal diseases pose a serious threat to global crop production and quality. Developing new and efficient fungicides is an important measure to control crop diseases.
Yao Tian, Jinchao Shi, Xiaoqian Deng, Tingyu Yu, Yong Hu, Richa Hu, Yufeng Lei, Linhua Yu, Xiang Zhu, Junkai Li   +9 more
doaj   +1 more source

Design and Synthesis In Silico Drug-like Prediction and Pharmacological Evaluation of Cyclopolymethylenic Homologous of LASSBio-1514

Molecules, 2021
Acylhydrazones are still an important framework to the design of new bioactive compounds. As treatment of chronic pain represents a clinical challenge, we decided to modify the structure of LASSBio-1514 (1), previously described as anti-inflammatory and ...
Lidia Moreira Lima, Tiago Fernandes da Silva, Carlos Eduardo da Silva Monteiro, Cristiane Aparecida-Silva, Walfrido Bispo Júnior, Aline Cavalcanti de Queiroz, Magna Suzana Alexandre-Moreira, Gisele Zapata-Sudo, Eliezer J. Barreiro   +8 more
doaj   +1 more source

‐Acylhydrazone

, 2022
Orthogonal chemistry is a valuable tool in the preparation of complex molecules as heteroglycoclusters. Unfortunately, selective heteroconjugation of multifunctional starting materials remains a usually challenging problem to overcome.
Fray, Marwa, Marwa Fray, David Lesur, Cragg, Peter, Mathiron, David, David Mathiron, Cragg, Peter; id_orcid, Rym Abidi, Serge Pilard, Abidi, Rym, Pilard, Serge, Benazza, Mohammed, Thouraya Barhoumi‐Slimi, Lesur, David, Mohammed Benazza, Frey, Marwa, Peter J. Cragg, Barhoumi-Slimi, Thouraya   +17 more
core   +1 more source

Design, Synthesis, and Bioactivities of Novel Tryptophan Derivatives Containing 2,5-Diketopiperazine and Acyl Hydrazine Moieties

Molecules, 2022
Based on the scaffolds widely used in drug design, a series of novel tryptophan derivatives containing 2,5-diketopiperazine and acyl hydrazine moieties have been designed, synthesized, characterized, and evaluated for their biological activities.
Lili Li, Rongxin Yang, Jianhua Liu, Jingjing Zhang, Hongjian Song, Yuxiu Liu, Qingmin Wang   +6 more
doaj   +1 more source

Design, synthesis and antifungal activity of novel 1,4-benzoxazin-3-one derivatives containing an acylhydrazone moiety

Frontiers in Chemistry, 2023
A series of 1,4-benzoxazin-3-one derivatives containing an acylhydrazone moiety were designed, synthesized and evaluated for their in vitro antifungal activities against Gibberella zeae, Pellicularia sasakii, Phytophthora infestans, Capsicum wilt, and ...
Chenghao Tang, Wenbo Guo, Shengzhou Yang, Xiuhong Hu, Xingju Chen, Xiang Wang   +5 more
doaj   +1 more source

3-Aminothiophene-2-Acylhydrazones: Non-Toxic, Analgesic and Anti-Inflammatory Lead-Candidates

Molecules, 2014
Different chemotypes are described as anti-inflammatory. Among them the N-acylhydrazones (NAH) are highlighted by their privileged structure nature, being present in several anti-inflammatory drug-candidates.
Yolanda Karla Cupertino da Silva, Christian Tadeo Moreno Reyes, Gildardo Rivera, Marina Amaral Alves, Eliezer J. Barreiro, Magna Suzana Alexandre Moreira, Lídia Moreira Lima   +6 more
doaj   +1 more source

New Palladacycle-Derived Acylhydrazones as Pre-catalysts in Mirozoki-Heck Coupling and Oxyarylations

Anais da Academia Brasileira de Ciências, 2018
New acylhydrazone-based palladacycles are prepared and evaluated as pre-catalysts in Mirozoki-Heck and oxyarylation reactions.
RAQUEL A.C. LEÃO, VAGNER D. PINHO, ARTUR S. COELHO, ARTHUR E. KÜMMERLE, PAULO R.R. COSTA   +4 more
doaj   +1 more source

Acylhydrazones as Widely Tunable Photoswitches

Journal of the American Chemical Society, 2015
Molecular photoswitches have attracted much attention in biological and materials contexts. Despite the fact that existing classes of these highly interesting functional molecules have been heavily investigated and optimized, distinct obstacles and inherent limitations remain.
Derk Jan van Dijken, † Petr Kovaříček, ‡ Svante P. Ihrig, and Stefan Hecht*   +3 more
openaire   +3 more sources

Synthesis, characterisation, conformational study and antibacterial activity of N-acylhydrazone and its derivatives [PDF]

, 2023
Researchers had examined N-acylhydrazone in great detail because of their pharmacological activities. For instance, N-acylhydrazone is found to be able to act as an antibacterial, anti-inflammatory, anticancer, anticonvulsant, antimalarial as well as ...
Tan, Yi Ying
core  

Synthesis and Spectral Characterization of Copper(II) and Zinc(II) Complexes of An Acylhydrazone [PDF]

, 2021
Copper(II) and zinc(II) complexes have been synthesized by the reaction of copper(II) acetate and zinc(II) acetate with an acylhydrazone and sodium cyanate and characterized by analytical and spectral ...
Vineetha, M C, Kurup, M R Prathapachandra   +1 more
core   +1 more source