Reactions of N-acylhydrazones with thionyl chloride [PDF]
Arkivoc, 2003 N-Acylhydrazones of o-hydroxyaryl ketones react with thionyl chloride to give Narylhydrazonoyl chlorides in good yields.
Antigoni Kotali, Ioannis S. Lafazanis
openaire +2 more sources
Química Nova, 2002 In this article are described new bioactive N-acylhydrazone (NAH) derivatives, structurally designed as optimization of aryl hydrazones precursors planned by molecular hybridization of two 5-lipoxigenase inhibitors, e.g. CBS-1108 and BW-755c.
Eliezer J. Barreiro +3 more
doaj +1 more source
Scientific African, 2023 Indole is an exceptional scaffold in the discovery and design of drugs with different mechanisms and biological activity. Numerous research has been conducted on N-acylhydrazones of indole and its derivatives, however, no account of the synthesis ...
Emmanuel Oloruntoba Yeye +3 more
doaj +1 more source
N′-[1-(Pyrazin-2-yl)ethylidene]pyrazine-2-carbohydrazide
IUCrData, 2018 The title compoud, C11H10N6O, was synthesized by the condensation reaction of pyrazine-2-carbohydrazide with 2-acetylpyrazine in ethanol. The dihedral angle between the pyrazine rings is 4.7 (3)°.
Zhaodong Wang
doaj +1 more source
Effects of MS-153 on chronic ethanol consumption and GLT1 modulation of glutamate levels in male alcohol-preferring rats [PDF]
, 2014 We have recently shown that upregulation of glutamate transporter 1 (GLT1) in the brain is associated in part with reduction in ethanol intake in alcohol-preferring (P) male rats. In this study, we investigated the effects of a synthetic compound, (R)-(−
Hasan Alhaddad +7 more
core +2 more sources
Synthesis, Spectroscopic characterization and invitro bacterial evaluation of Ni(II) complexes of new tridentate aroylhydrazone ligands [PDF]
, 2016 Nickel(II) complexes of four new aroylhydrazones,N-(2-hydroxy-1-naphthaldehyde)- N\u27 -(4-nitrobenzoyl)hydrazone(H2L1), N-(2-hydroxy-4-methoxybenzaldehyde)-N\u27-(2-furoyl) hydrazone (H2L2), N-(2-hydroxyacetophenone)-N\u27 -(2-theonyl) hydrazone (H2L3 ...
Banerjee, K. (Kamalika) +2 more
core +1 more source
Chiral Assembly Preferences and Directing Effects in Supramolecular Two-Component Organogels [PDF]
, 2018 The impact of chirality on the self-assembly of supramolecular gels is of considerable importance, as molecular-scale programming can be translated into nanostructuring and ultimately affect macroscopic performance.
Edwards, William, Smith, David Kelham
core +5 more sources
Global Challenges, 2019 Gel adsorbents are promising for pollutant removal from the wastewater. Herein, an acylhydrazone gel is developed from acylhydrazide‐terminated pentaerythritol (PAT) and 2,4,6‐triformylphloroglucinol (TFP) based on dynamic covalent acylhydrazone ...
Haobin Fang +4 more
doaj +1 more source
Design, Synthesis, Antinociceptive and Anti-Inflammatory Activities of Novel Piroxicam Analogues
Molecules, 2012 In this paper we report the design, synthesis, antinociceptive and anti-inflammatory activities of a series of benzothiazine N-acylhydrazones 14a–h, planned by structural modification of piroxicam (1), a non steroidal anti-inflammatory drug ...
Eliezer J. Barreiro +8 more
doaj +1 more source
Isoenzyme- and Allozyme-Specific Inhibitors: 2,20-Dihydroxybenzophenones and Their Carbonyl N-Analogues that Discriminate between Human Glutathione Transferase A1-1 and P1-1 Allozymes [PDF]
, 2015 The selectivity of certain benzophenones and their carbonyl N-analogues was investigated towards the human GSTP1-1 allozymes A, B and C involved in MDR. The allozymes were purified from extracts derived from E.
Clonis, Yannis D. +5 more
core +1 more source