Bicyclic amido compounds with antiprotozoal activity
Aroyl derivatives of 2-aminobicyclo-octanes and 2-azabicyclo-nonanes have been synthesized and tested for their activities against the causative organisms of East African trypanosomiasis and malaria tropica.
Brun, R. +5 more
core
Synthesis and antiprotozoal activity of some imidazoles derivatives
The synthesis and in vitro antiprotozoal activity of a series of nitroimidazoles are described. A substituted phenyl group and, in many of the compounds, a N-substituent were also present: vinylogues of some of the compounds are described. Several of the
L Golberg +4 more
core +1 more source
Synthesis, antiprotozoal and antibacterial activity of nitro- and halogeno-substituted benzimidazole derivatives [PDF]
Two series of benzimidazole derivatives were sythesised. The first one was based on 5,6-dinitrobenzimidazole, the second one comprises 2-thioalkyl- and thioaryl-substituted modified benzimidazoles. Antibacterial and antiprotozoal.
Upcroft, Jacqueline +6 more
core +1 more source
Antiprotozoal Sesquiterpene Pyridine Alkaloids from Maytenus ilicifolia
As part of a bioprospecting program aimed at the discovery of antiprotozoal agents from the Brazilian flora, two new sesquiterpene pyridine alkaloids, ilicifoliunines A (1) and B (2), along with the known alkaloids aquifoliunine E-I (3) and mayteine (4),
Nogueira, Claudio R. [UNESP] +17 more
core +1 more source
Antiprotozoal activity of synthetic amino substituted 1-methyl-1H-
: The antiprotozoal properties of a series of amino substituted 1-methyl-1H--carbolines were investigated in a broad panel of parasites. Various substituents were systematically introduced at various positions on the carbocyclic ring of the parent 1 ...
Yadav, Ashok Kumar +7 more
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Antiprotozoal and antiangiogenic saponins from **Apodytes dimidiata**
: Bioassay-guided isolation was performed on the leaves of Apodytes dimidiata E. Mey. Ex Arn. (Icacinaceae), based on previously demonstrated activity against Leishmania.
Cuyckens, Filip +6 more
core
Brazilian <i>Bothrops</i> and <i>Crotalus</i> Snake Venoms as a Source of Antiprotozoal Agents: Unlocking Toxins for Therapeutic Development. [PDF]
Reis TC +8 more
europepmc +1 more source
Molecular epidemiology and risk factors associated with Babesia bigemina infection in cattle. [PDF]
Selim A +6 more
europepmc +1 more source
Perovskone, a potential antiprotozoal hit compound, quantification and derivatization. [PDF]
Kamelan Zargar Zarin M +7 more
europepmc +1 more source
Editorial: Drug Re-purposing for the Treatment of Bacterial and Viral Infections
Rodolfo García-Contreras +2 more
doaj +1 more source

