Continuous-Flow Hofmann Rearrangement Using Trichloroisocyanuric Acid for the Preparation of 2-Benzoxazolinone [PDF]
, 2022 A continuous-flow preparation of 2-benzoxazolinone via the Hofmann rearrangement of salicylamide has been implemented employing trichloroisocyanuric acid as the stable and atom-economic chlorinating agent.
Baxendale, Ian R., Gambacorta, Guido
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Biochemical interaction of twenty steroid derivatives with ribosomal protein kinase 4 S6 (RSK-4) surface using a theoretical model [PDF]
, 2023 Several genetic expressions have been involved in the development of cancer such as the expression of a ribosomal kinase S6 P90 (RSK-4). It is important to mention that some compounds such as LJH685, 2073047-06-8, and SL0101 can act as RSK-4 inhibitors ...
Alvarez-Ramirez, Magdalena +8 more
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Synthesis of enamines and their bromination [PDF]
, 2011 Enamines represent an important class of reactive intermediates in organic synthesis. They are frequently used as a potential building block to access several types of heterocyclic ring systems and biologically active analogues.
Thakur, Vasundhara
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Mechanisms of growth inhibition of Phytomonas serpens by the alkaloids tomatine and tomatidine [PDF]
, 2015 Phytomonas serpens are flagellates in the family Trypanosomatidae that parasitise the tomato plant (Solanum lycopersicum L.), which results in fruits with low commercial value.
Beach DH +47 more
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Design and synthesis of novel Azasteroids and Pseudoazulenyl nitrones [PDF]
, 2016 Steroids are one of the essential classes of bioactive compounds and are involved in many biological functions which include their role as signaling compounds, the alteration of membrane fluidity and the regulation of a variety of metabolic processes. In
Birudukota, Nagaraju
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Advances in the development of hybrid anticancer drugs [PDF]
, 2013 Introduction: Hybrid anticancer drugs are of great therapeutic interests as they can potentially overcome most of the pharmacokinetic drawbacks encountered when using conventional anticancer drugs.
Bérubé, Gervais, Fortin, Sébastien
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Insecticides Based on Differences in Metabolic Pathways [PDF]
, 1990 Insects have been major pests of humankind at least since the beginning of recorded history. To this day insects continue to cause problems in domestic, agricultural, and health situations.
Cunningham, G N. +2 more
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Acyl radical cascade reactions: the synthesis of azasteroids [PDF]
, 1998 Our work has been concerned with the synthesis of azasteroid ring systems, utilising acyl radical cascade reactions. Chapter 1 comprises an overview of published work relevant to our studies: an analysis of steroid biosynthesis and synthesis; a review of
Double, Philip John
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Studies on The Synthesis of B-Ring 6-Azasteroids [PDF]
, 2006 Azasteroids, which carry a nitrogen in the C-6 position of the steroid nucleus are still mysterious and very few synthesized, were found to possess antimicrobial and antifungal properties apart from their pharmacodynamic actions. The literature reports
Gandikota, Jyothi
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Synthesis and molecular docking of 2,4,5-trisubstituted- 1,3-thiazole derivatives as antibacterial agents = Sintesis dan penyatuan molekul terbitan 1,3-tiazol berpenggantian-2,4,5 sebagai agen antibakteria [PDF]
, 2019 The emergence of antibiotic resistance against bacterial strains has attracted great interest in the discovery and development of new antibacterial agents. Thiazole derivatives have been widely used in the biological as well as pharmacological fields and
Abdullah Ripain, Iswatun Hasanah +5 more
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