Results 21 to 30 of about 1,295 (195)

The synthesis of 9-azasteroids—II

open access: yesTetrahedron, 1965
Abstract The synthesis of 3-cyano-4-oxo-1,2,3,4,5,6-hexahydrobenzo[c]quinolizine (XIV), of 2-carbethoxy-3-oxo-1,2,3,4,5,6-hexahydrobenzo[c]quinolizine(XVII), and of 4-cyano-3-oxo-1,2,3,4,5,6-hexahydrobenzo[c]quinolizine (XXIX) is reported. Attempts to methylate 3-carbethoxy-4-oxo-1,2,3,4,5,6-hexahydrobenzo[c]quinolizine (II) were unsuccessful ...
G. Jones, J. Wood
openaire   +2 more sources

Azasteroids—VI

open access: yesTetrahedron, 1967
A.I. Meyers, J.C. Sircar
openaire   +2 more sources

The Mce3R Regulon Is Required for 6-Azasteroid Potentiation of Anti-TB Drug Activity [PDF]

open access: green, 2018
Cholesterol is important for Mycobacterium tuberculosis (Mtb) survival and persistence in the host. We describe a series of 6-azasteroids tested as cholesterol analogs, that are synergistic inhibitors of Mtb viability.
Xinxin Yang   +4 more
openalex   +2 more sources

19-Nor-10-azasteroids:  A Novel Class of Inhibitors for Human Steroid 5α-Reductases 1 and 2

open access: greenJournal of Medicinal Chemistry, 1997
Antonio Guarna   +11 more
openalex   +2 more sources

Design, Synthesis, and Biological Evaluation of 16-Substituted 4-Azasteroids as Tissue-Selective Androgen Receptor Modulators (SARMs)

open access: greenJournal of Medicinal Chemistry, 2009
Helen J. Mitchell   +16 more
openalex   +2 more sources

The synthesis of 2-azasteroids

open access: yesTetrahedron Letters, 1972
Raphael Pappo, Robert J. Chorvat
openaire   +2 more sources

4,7.beta.-Dimethyl-4-azacholestan-3-one (MK-386) and Related 4-Azasteroids as Selective Inhibitors of Human Type 1 5.alpha.-Reductase

open access: greenJournal of Medicinal Chemistry, 1994
Raman K. Bakshi   +9 more
openalex   +2 more sources

Effect of Dietary Azasteroids on the Growth and Development of the Gram Pod Borer Helicoverpa armigera (Hubner)

open access: yesIndian Journal of Entomology, 2022
Effect of two azasteroids, 25-azacholestane and 25-azacoprostane was studied on growth and development of an economically important phytophagous pest, Helicoverpa armigera (Hubner) causing extensive damage to crops like cotton, pigeon pea, chickpea and ...
Rita Rath   +3 more
semanticscholar   +1 more source

Azasteroids: structure-activity relationships for inhibition of 5.alpha.-reductase and of androgen receptor binding

open access: greenJournal of Medicinal Chemistry, 1986
Gary H. Rasmusson   +9 more
openalex   +2 more sources

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