Skeletal Editing via Diastereoselective Ring Expansion Enables Enantioenriched Tetrasubstituted Δ<sup>3</sup>‑Oxepenes. [PDF]
Naulin E +3 more
europepmc +1 more source
Site-Selective C6-β-Aminoalkylation of Tetrahydroquinolines with N-Arylsulfonyl Aryl Aziridines in Hexafluoroisopropanol: A Modular Approach to C6-Alkylated Quinolines. [PDF]
Taskesenligil Y, Aslan M, Saracoglu N.
europepmc +1 more source
Synthesis of an N-Galactosyl Norbornane Aziridine and its Potent Mixed Inhibition of Aspergillus oryzae β-Galactosidase. [PDF]
McCormack A, Gavin R, Bols M, Murphy PV.
europepmc +1 more source
Iodonitrene-Mediated Nitrogen Transfer to Alkenes for the Direct Synthesis of NH-Aziridines. [PDF]
Gelato Y +7 more
europepmc +1 more source
Two-carbon ring expansion of bicyclic aziridines to oxazocines <i>via</i> aryne insertion into a σ C-N bond. [PDF]
Rampon DS +7 more
europepmc +1 more source
Photocatalyzed Ring Expansion of α-Ketosulfonylaziridines: Ready Access to δ-Sultams. [PDF]
Mastandrea MM +7 more
europepmc +1 more source
Aziridine - Triazole Conjugates as a Novel Class of MMP-2 Inhibitors
We report here the synthesis of a series of (aryltriazolyl)methylaziridines 1 and their evaluation as selective inhibitors of MMP-2.[2] They constitute a novel class of hydroxamic acid-free matrix metalloproteinase ...
Romanchikova, Nadezhda +3 more
core
Synthesis and Application of Bioactive N-Functionalized Aziridines. [PDF]
Tan H +4 more
europepmc +1 more source
Cascade transformation of 2-(diazoacetyl)-2<i>H</i>-azirines to 2-aroyl-3-hydroxy-1<i>H</i>-pyrroles via condensation with aromatic aldehydes. [PDF]
Zanakhov TO +3 more
europepmc +1 more source
Sulfenate anion catalyzed enantio- and diastereoselective aziridination. [PDF]
Pu Y, Smaldone AM, Adrio J, Walsh PJ.
europepmc +1 more source

