Transition Metal-Catalyzed Synthesis and Reactivity of N-Alkenyl Aziridines
Straightforward methods for palladium-catalyzed alkenylation of aziridines with alkenyl halides and copper-catalyzed alkenylation of aziridines with alkenyl boronic acids have been developed.
Shadi Dalili (2689783) +1 more
core +1 more source
Solvent- and Temperature-Dependent Functionalization of Enantioenriched Aziridines
A highly stereo- and regioselective functionalisation of chiral nonracemic aziridines is reported. By starting from a parent enantioenriched aziridine and finely tuning the reaction conditions, it is possible to address the regio- and ...
M. C, MUSIO +7 more
core +1 more source
Development and application of the vinylepoxide – dihydrofuran rearrangement [PDF]
The vinylepoxide - diliydrofuran rearrangement offers a route to substituted 2,3- dihydrofurans with a high degree of diastereoselectivity. The rearrangement proceeds via an ylide-type intermediate arising from the thermolysis of a carbon-carbon epoxide ...
Dutton, William Martin
core
Enantio- and regioselective nickel/photoredox-catalyzed cross-electrophile coupling of benzylic aziridines with alkynyl bromides. [PDF]
Lan H +4 more
europepmc +1 more source
Adapting Bower's intramolecular aziridination reaction allows for a metal-free synthesis of N-H aziridines. [PDF]
Silver R, Kelley SP, Sathyamoorthi S.
europepmc +1 more source
Oseltamivir aziridines are potent influenza neuraminidase inhibitors and imaging agents. [PDF]
Vriends MBL +22 more
europepmc +1 more source
Site-Selective C6-β-Aminoalkylation of Tetrahydroquinolines with N-Arylsulfonyl Aryl Aziridines in Hexafluoroisopropanol: A Modular Approach to C6-Alkylated Quinolines. [PDF]
Taskesenligil Y, Aslan M, Saracoglu N.
europepmc +1 more source
Bifunctional Aziridines from Photochemically Generated FSO<sub>2</sub>NH<sub>2</sub> for SuFEx Diversification of Alkenes. [PDF]
Choudhury A +3 more
europepmc +1 more source
Stereofacial Assembly of Engineered Multichiral Aziridines via B/Si Ylide Insertion. [PDF]
Pujol M +4 more
europepmc +1 more source
A Polarity-Mismatched Photocatalytic Cross-Coupling Enables Diversity-Oriented Synthesis of aza-Heterocycles. [PDF]
Urbańczyk J +5 more
europepmc +1 more source

