Results 61 to 70 of about 38,481 (291)

The 68Ga-labeled chlorinated benzamide derivative: A novel PET imaging probe for detection of melanoma

Results in Chemistry
The benzamide structure is known for its ability to target melanin, a specific biomarker of melanoma. Therefore, we developed a new chlorinated benzamide structure for the detection of melanoma on positron emission tomography (PET). The derived benzamide
Yejin Seo, Dagyeong Hong, Eunsu Kim, Chaewon Lee, Boreum Song, Wookyeong Jeong, Jiyu Kim, Seong-Young Kwon, Dong-Yeon Kim, Ayoung Pyo   +9 more
doaj   +1 more source

Crystal structure of 3-chloro-N-(2-nitrophenyl)benzamide

Acta Crystallographica Section E: Crystallographic Communications, 2015
In the title compound, C13H9ClN2O3, the mean plane of the central amide fragment (r.m.s. deviation = 0.016 Å) subtends dihedral angles of 15.2 (2) and 8.2 (2)° with the chloro- and nitro-substituted benzene rings, respectively.
Rodolfo Moreno-Fuquen, Alexis Azcárate, Alan R. Kennedy   +2 more
doaj   +1 more source

3,5-Dibromo-4-carbamoylbenzoic acid 2-propanol monosolvate

IUCrData, 2021
In the title solvated crystal, C8H5Br2NO3·C3H8O, the acid molecules form inversion dimers by pairwise N—H...O hydrogen bonds between carbamoyl groups and the carboxyl and carbamoyl groups link to form head-to-tail inversion dimers.
Wayland E. Noland, Ryan J. Herzig, Renee J. Fox, Kenneth J. Tritch   +3 more
doaj   +1 more source

Synthesis and characterisation of a new benzamide-containing nitrobenzoxadiazole as a GSTP1-1 inhibitor endowed with high stability to metabolic hydrolysis [PDF]

, 2019
The antitumor agent 6-((7-nitrobenzo[c][1,2,5]oxadiazol-4-yl)thio)hexan-1-ol (1) is a potent inhibitor of GSTP1-1, a glutathione S-transferase capable of inhibiting apoptosis by binding to JNK1 and TRAF2.
Caccuri, A. M., De Luca, A., Di Paolo, V., Fulci, C., Lucidi, A., Morozzo Della Rocca, B., Quintieri, L., Rosato, A., Rotili, D., Sciarretta, F.   +9 more
core   +2 more sources

Piezofluorochromism in Aramid Dyads: Pressure‐Triggered Luminescence Enhancement with Predictable Emission Shifts

Advanced Science, EarlyView.
High‐pressure investigations uncover the structural determinants of luminescence intensity and shifts in aramids, establishing intrinsic intramolecular rotation as a reliable predictor of their piezofluorochromic behavior. Leveraging this insight, conjugation modulation is proposed as a precise strategy to tune their piezofluorochromic properties ...
Yayun Wang, Zhe Jia, Yaru Wang, Lin Wei, Zimin Hao, Yanan Wang, Jingwen Guo, Aisen Li, Lei Li, Kai Wang, Qian Li   +10 more
wiley   +1 more source

Enhancing the cellular uptake of Py–Im polyamides through next-generation aryl turns [PDF]

, 2012
Pyrrole–imidazole (Py–Im) hairpin polyamides are a class of programmable, sequence-specific DNA binding oligomers capable of disrupting protein–DNA interactions and modulating gene expression in living cells.
Baird, Belitsky, Best, Bijsterbosch, Bradford, Chenoweth, Chenoweth, Chenoweth, Cleutjens, Cohen, Crowley, David C. Montgomery, Dervan, Dervan, Dickinson, Dose, D’Adamio, Edelson, Edwards, Gissot, Herman, Hesselberth, Hsu, Hsu, Jacobs, Johnson, Jordan L. Meier, Krutzik, Kwon, Magee, Mapp, Matsuda, Meijsing, Mrksich, Muzikar, Nickols, Nickols, Nickols, Nishijima, Ohtsukia, Olenyuk, Peter B. Dervan, Poulin-Kerstien, Reddy, Riegman, Rucker, Schmidt, Schultz, So, Swalley, Tsai, Van Dyke, Vaquerizas, Vichai, Yao   +54 more
core   +2 more sources

68Ga-labeled fluorinated benzamide derivatives for positron emission tomography imaging of melanoma. [PDF]

PLoS One
Lee C, Song B, Kim E, Seo Y, Hong D, Kim J, Jeong W, Kwon SY, Kim DY, Pyo A.   +9 more
europepmc   +3 more sources

Performance of the ALOGPS 2.1 program for octanol-water partition coefficient prediction with organic chemicals on the Canadian Domestic Substances List [PDF]

, 2010
The KOWWIN and ALOGPS octanol-water partition coefficient (K~ow~) estimation software programs were compared for their capacity to accurately predict log K~ow~ values of 1545 organic compounds on the publicly available Domestic Substances List (DSL) from
Kaya Forest, Sierra Rayne
core   +2 more sources

The development of a micro technique for qualitative organic analysis [PDF]

, 1934
Thesis (M.A.)--Boston ...
Rapport, Arthur
core   +1 more source

para-Selective C-H amidation of simple arenes with nitriles [PDF]

, 2015
A para-selective C-H amidation of simple arenes with nitriles has been developed. By increasing the amount of arenes, a further meta-selective C-H arylation of the produced amides occurred.
Allen, Allen, Antonchick, Casitas, Chen, Fañanás-Mastral, Gao, Grohmann, Guérinot, Harvey, He, He, Hsieh, Huffman, Ichiishi, Ichiishi, Kantak, Kawano, Kim, Kim, King, Li, Li, Louillat, Lv, Marchetti, Matsuda, Nadres, Ng, Ng, Ng, Ng, Peng, Phipps, Phipps, Pialat, Ryu, Ryu, Shai, Shin, Shrestha, Skucas, Sokolovs, Su, Tew, Thomas, Thu, Tran, Tsang, Valeur, Wang, Wang, Wang, Xiang, Xu, Yoo, Zhang, Zhang, Zhang, Zhao   +59 more
core   +2 more sources