Results 161 to 170 of about 2,089 (211)

Development of human growth hormone-treated chimeric mice with humanized livers for an evaluation model of drug-induced fatty liver disease. [PDF]

Arch Toxicol
Morioka S, Sanoh S, Ishida Y, Furukawa S, Ogawa Y, Kotake Y, Tateno C.   +6 more
europepmc   +1 more source

Synthesis, in vitro evaluation and computational modelling of benzene sulfonamide derivatives as Dickkopf 1 inhibitors for anticancer drug development. [PDF]

Sci Rep
Bilal MS, Ejaz SA, Naseem S, Channar PA, Saeed A, Zargar S, Ujan R, Sahito R, Abbas Q, Wani TA.   +9 more
europepmc   +1 more source

A general strategy for high-efficiency live bacteria imaging and targeted phototherapy. [PDF]

Chem Sci
Wang X, Ding L, Liu J, Lv J, Liu J, Yan Y, Li X, Shi H, Wang H, Wang J, Liu S, Cao D, Yang X, Xue L.   +13 more
europepmc   +1 more source

Novel Derivatives of 3-Amino-4-hydroxy-benzenesulfonamide: Synthesis, Binding to Carbonic Anhydrases, and Activity in Cancer Cell 2D and 3D Cultures. [PDF]

Int J Mol Sci
Vainauskas V, Norvaišaitė R, Grybaitė B, Vaickelionienė R, Smirnov A, Kojis T, Baranauskiene L, Manakova E, Gražulis S, Zubrienė A, Matulis D, Mickevičius V, Petrikaitė V.   +12 more
europepmc   +1 more source

Revisiting the Effect of Udenafil on Exercise Performance in Patients With Fontan Circulation: Results of a Post Hoc Analysis of the FUEL Trial. [PDF]

J Am Heart Assoc
Goldberg DJ, Zak V, Hu C, Lubert AM, Rathod RH, Penny DJ, Whitehill R, Schumacher KR, Ginde S, Ploutz M, Kim GB, Nowlen TT, DiMaria MV, Frischhertz BP, Wagner JB, McHugh KE, McCrindle BW, Cartoski MJ, Detterich J, Yetman AT, John AS, Richmond ME, Files M, Payne RM, Mackie AS, Davis CK, Orr WB, Garg R, Hill KD, Yauck JS, McBride MG, Yeager J, Pearson GD, Paridon SM, Goldstein BH.   +34 more
europepmc   +1 more source

Selective phosphoinositide 3-kinase inhibitors and implication in diabetic retinopathy as pharmacological tools. [PDF]

Front Pharmacol
Bonaccorso C, Lazzara F, La Rosa I, Munzone C, Grasso A, Platania CBM, Bucolo C.   +6 more
europepmc   +1 more source

Synthesis and carbonic anhydrase inhibitory activities of new thienyl-substituted pyrazoline benzenesulfonamides

Journal of Enzyme Inhibition and Medicinal Chemistry, 2016
A series of new thienyl-substituted pyrazoline benzenesulfonamides were synthesized and their carbonic anhydrase (CA, EC 4.2.1.1) inhibitory activities were tested on the human (h) isoforms hCA I and hCA II.
Ebru Mete, Birnur Comez, Halise Inci Gul   +2 more
exaly   +2 more sources

Design, synthesis and biological evaluation of novel ureido benzenesulfonamides incorporating 1,3,5-triazine moieties as potent carbonic anhydrase IX inhibitors

Bioorganic Chemistry, 2019
A series of novel ureido benzenesulfonamides incorporating 1,3,5-triazine moieties were obtained by reacting 4-isocyanato-benzenesulfonamide (2) with 2-amino-4,6-dicholoro-1,3,5-triazine (4).
Nebih Lolak, Suleyman Akocak, Silvia Bua   +2 more
exaly   +2 more sources

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Pharmacophoric 2-hydroxyalkyl benzenesulfonamide: A single-step synthesis from benzenesulfonamide via hemiaminal

European Journal of Medicinal Chemistry, 2007
ortho-Acylation attempt of benzenesulfonamide afforded the corresponding hemiaminal as major product. The in situ reduction of the reaction mixture, reported herein, directly provided 2-hydroxyalkyl benzenesulfonamide, an important pharmacophoric element for designing drug-like scaffolds. Its application is demonstrated through designing a novel series
Sunil K, Singh, S, Shivaramakrishna, V, Saibaba, K Srinivas, Rao, K Ravi, Ganesh, R, Vasudev, P Praveen, Kumar, J Moses, Babu, K, Vyas, Y Koteswar, Rao, J, Iqbal   +10 more
openaire   +3 more sources

Synthesis of benzenesulfonamide serinol by the Hinsberg reaction

Ministry of Science and Technology, Vietnam, 2022
This research focused on synthesising benzenesulfon-amide serinol (BSSe), a new sulfonamide monomer, by the Hinsberg reaction between primary amine of serinol and sulfonyl of benzenesulfonyl chloride (BSC) in an al-kaline environment. The effect of the reacted environ-ment on the reaction efficiency and structure of BSSe were investigated.
Vu Viet Linh Nguyen, Thi Xuan Thao Tran, Ngoc Tan Nguyen, Dai Phu Huynh   +3 more
openaire   +1 more source