Results 121 to 130 of about 9,350 (208)

Synthesis, Characterization, and Biological Evaluation of Aliphatic-Substituted Benzimidazole Derivatives: Induction of Apoptosis, Cell Cycle Arrest, and Molecular Docking in Breast Cancer Cells. [PDF]

Drug Dev Res
Keser M, Çamlı Pulat Ç, Atmaca H, Akgün H, Albay C, Menteşe E, Bektaş H, Ilhan S.   +7 more
europepmc   +1 more source

Virtual Screening of Benzimidazole Derivatives as Potential Triose Phosphate Isomerase Inhibitors with Biological Activity against Leishmania mexicana. [PDF]

Pharmaceuticals (Basel), 2023
Vázquez-Jiménez LK, Juárez-Saldivar A, Chan-Bacab MJ, Delgado-Maldonado T, González-Morales LD, Palos I, Ortiz-Pérez E, Lara-Ramírez EE, Ramírez-Moreno E, Rivera G.   +9 more
europepmc   +1 more source

Searching for Novel COVID19 Treatments: Towards Covalent TMPRSS2 Inhibitors

ChemMedChem, Volume 21, Issue 19, 14 October 2026.
We designed, synthesised, and evaluated new guanidine derivatives as potential covalent inhibitors of TMPRSS2, a key protease for SARS‐CoV‐2 entry. Computational studies showed that some compounds have improved binding over nafamostat. However, experimentally none effectively blocked viral entry in cell assays, indicating further optimisation is needed.
Marco Minneci, Barbara Farkaš, Adeyemi Rahman, Inga Nehlmeier, Amy Eichmann, Stefan Pöhlmann, Isabel Rozas   +6 more
wiley   +1 more source

Synthesis of piperazine-based benzimidazole derivatives as potent urease inhibitors and molecular docking studies. [PDF]

Sci Rep
Shahriarynejad D, Dastyafteh N, Naz F, Talebi M, Safapoor S, Ghafouri SN, Azizian H, Mohammadi-Khanaposhtani M, Larijani B, Asadi M, Amanlou M, Mahdavi M, Khan KM.   +12 more
europepmc   +1 more source

Fighting Antibiotic Resistance: New Pyrimidine-Clubbed Benzimidazole Derivatives as Potential DHFR Inhibitors. [PDF]

Molecules, 2023
Haque MA, Marathakam A, Rana R, Almehmadi SJ, Tambe VB, Charde MS, Islam F, Siddiqui FA, Culletta G, Almerico AM, Tutone M, Khan SL.   +11 more
europepmc   +1 more source

Dual Porphyrin Sensitized Photocatalytic System for Visible‐Light‐Driven CO2 Reduction

ChemSusChem, Volume 19, Issue 19, 14 October 2026.
Dual porphyrin–sensitized TiO2 enables efficient visible‐light CO2 reduction by integrating Zn‐porphyrin photosensitization with urea‐functionalized Fe‐porphyrin catalysts. Immobilization enhances charge separation, activity, and durability, while tuning electron donor and proton availability reveals key aspects that influence this catalytic conversion.
Anna Katsari, Emmanouil Nikoloudakis, Georgios Charalambidis, Antonios Iliakis, Fabrice Odobel, Emmanuel Stratakis   +5 more
wiley   +1 more source

Comment on "Influence of Solvents and Halogenation on ESIPT of Benzimidazole Derivatives for Designing Turn-on Fluorescence Probes". [PDF]

ACS Omega
Nedeltcheva-Antonova D, Antonov L.
europepmc   +1 more source

Design, Synthesis, and Characterization of Novel Coordination Compounds of Benzimidazole Derivatives with Cadmium. [PDF]

Pharmaceutics, 2022
Raducka A, Świątkowski M, Korona-Głowniak I, Kaproń B, Plech T, Szczesio M, Gobis K, Czylkowska A.   +7 more
europepmc   +1 more source

Evaluation of the Antileishmanial Activity of Some Benzimidazole Derivatives Using In Vitro and In Silico Techniques. [PDF]

Vet Sci
Eser M, Çavuş İ, Kaya AZ, Evren AE, Yurttaş L.   +4 more
europepmc   +1 more source

Reply to the Comment on "Influence of Solvents and Halogenation on ESIPT of Benzimidazole Derivatives for Designing Turn-on Fluorescence Probes". [PDF]

ACS Omega
Queiroz MH, Nascimento JL, Alves TV, Rivelino R, Canuto S.   +4 more
europepmc   +1 more source