Results 41 to 50 of about 547 (150)

Cardiovascular activity of 1,2,4-benzothiadiazine-1,1-dioxide derivatives Part 10

open access: yes, 1988
The Ms deals with the synthesis and in vivo activity of a series of benzothiadiazines as cardiovascular ...
PARENTI, Carlo   +4 more
core  

Structures of SUR2 NBD1 / Drug Complexes Determined with NMR Spectroscopy and Data Driven Docking

open access: yes, 2021
ATP-sensitive potassium (KATP) channels are formed by four inward-rectifying K+ channels and four regulatory sulfonylurea receptors (SURs). ATP binding and hydrolysis at the SUR nucleotide binding domains (NBDs) regulates opening of the KATP channel pore.
Sayewich, Jonathan Scott
core  

Heteroarylalkanoic acids with possible antiinflammatory activities. Note IV

open access: yes, 1987
The Ms deals with the synthesis and in vivo activity of a series of benzothiadiazines as potential nonsteroidal antiinflammatory ...
PARENTI, Carlo   +5 more
core  

A short, versatile route towards benzothiadiazinyl radicals. [PDF]

open access: yesChem Sci, 2021
Borys AM   +4 more
europepmc   +1 more source

5-Arylbenzothiadiazine Type Compounds as Positive AllostericModulators of AMPA/Kainate Receptors

open access: yes, 2012
The potential therapeutic benefit of compounds able to activate AMPA receptors (AMPAr) has led to the search for new AMPAr positive modulators. On the basis of crystallographic data of the benzothiadiazines binding mode in the S1S2 GluA2 dimer ...
C. PARENTI   +10 more
core   +2 more sources

5-Arylbenzothiadiazine Type Compounds as Positive Allosteric Modulators of AMPA/Kainate Receptors

open access: yes, 2016
The potential therapeutic benefit of compounds able to activate AMPA receptors (AMPAr) has led to the search for new AMPAr positive modulators. On the basis of crystallographic data of the benzothiadiazines binding mode in the S1S2 GluA2 dimer interface,
Umberto M. Battisti (2127295)   +10 more
core   +1 more source

In silico identification of promising inhibitor against RNA-dependent RNA polymerase target of SARS-CoV-2. [PDF]

open access: yesMol Biol Res Commun, 2021
Singh P   +4 more
europepmc   +1 more source

The action of diazoxide analogs on aortic reactivity in normotensive and spontaneously hypertensive rats

open access: yes, 1977
Diazoxide and four related 1,2,4-benzothiadiazines reduced the maximum responses to noradrenaline (NA) and KCl in aortic rings from normotensive and spontaneously hypertensive rats (SHR).
S. Chona, D. J. Triggle
core   +1 more source

Heteroarylalkanoic acids with possiblre antiinflammatory activities. Note V. The scavenging of the oxygen free-radicals

open access: yes, 1988
The Ms deals with the determination of the free radicals scavenging ability of a series of benzothiadiazines provided with antiinflammatory ...
PARENTI, Carlo   +3 more
core  

New derivatives of 1,2,4-benzothiadiazines and their coordination chemistry

open access: yes, 2018
Chapter 1 provides an introduction to coordination chemistry and polydentate N-donor ligands along with a synopsis of heterocycles with N and S/N donor atoms.
Pringouri, Konstantina
core  

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