Synthesis and Antimicrobial Activity of 1,2-Benzothiazine Derivatives [PDF]
Molecules, 2016 A number of 1,2-benzothiazines have been synthesized in a three-step process. Nine chalcones 1–9 bearing methyl, fluoro, chloro and bromo substituents were chlorosulfonated with chlorosulfonic acid to generate the chalcone sulfonyl chlorides 10–18. These
Chandani Patel +6 more
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Efficient synthesis of benzothiazine and acrylamide compounds [PDF]
Química Nova, 2010 This article describes the synthesis of the new (2Z)-2-(4-methoxybenzylidene)-6-nitro-4H -benzo[1,4]thiazin-3-one, (2Z)-2-(4-methoxybenzylidene)-4-methyl-6-nitro-4H-benzo[1,4]thiazin-3-one, (2Z)-6-amino-2-(4-methoxybenzylidene)-4H -benzo[1,4]thiazin-3 ...
Ana Maria Alves Souza +8 more
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Evaluation of 1,2-Benzothiazine 1,1-Dioxide Derivatives In Vitro Activity towards Clinical-Relevant Microorganisms and Fibroblasts [PDF]
Molecules, 2020 The global concern related with growing number of bacterial pathogens, resistant to numerous antibiotics, prone scientific environment to search for new antimicrobials.
Ruth K. Dudek-Wicher +5 more
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Potential anti-amoebic effects of synthetic 1,4-benzothiazine derivatives against Acanthamoeba castellanii [PDF]
HeliyonA rare but lethal central nervous system disease known as granulomatous amoebic encephalitis (GAE) and potentially blinding Acanthamoeba keratitis are diseases caused by free-living Acanthamoeba.
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Methyl 4-ethoxy-2-methyl-2H-1,2-benzothiazine-3-carboxylate 1,1-dioxide [PDF]
Acta Crystallographica Section E, 2008 In the crystal structure of the title compound, C13H15NO5S, the molecules exhibit weak S=O...H—C and C=O...H—C intermolecular interactions and arrange themselves into centrosymmetric dimers by means of π–π interactions (ring ...
Muhammad Zia-ur-Rehman +4 more
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N-(3,4-Dimethylphenyl)-4-hydroxy-2-methyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide [PDF]
Acta Crystallographica Section E, 2009 1,2-Benzothiazines similar to the title compound, C18H18N2O4S, are well known in the literature for their biological activities and are used as medicines in the treatment of inflammation and rheumatoid arthritis. The thiazine ring adopts a distorted half-
Waseeq Ahmad Siddiqui +4 more
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Enantioselective reduction of sulfur-containing cyclic imines through biocatalysis. [PDF]
Nat Commun, 2018 Zumbrägel N, Merten C, Huber SM, Gröger H. Enantioselective reduction of sulfur-containing cyclic imines through biocatalysis. Nature Communications.
Zumbrägel N +3 more
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Heterocyclic Electrochemistry: Renewable Electricity in the Construction of Heterocycles. [PDF]
ACS Omega, 2023 Numerous applications in the realm of biological exploration and drug synthesis can be found in heterocyclic chemistry, which is a vast subject. Many efforts have been developed to further improve the reaction conditions to access this interesting family
Aslam S +5 more
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Synthesis of Anthraquinone Mono- and Diboron Complexes with Near-Infrared Panchromatic Absorption. [PDF]
ChemistryAnthraquinone boron complexes bearing β‐iminoenolate ligand(s) exhibit strongly substituent‐dependent absorption properties. Unsubstituted monoboron and diboron complexes show sharp UV–Vis–NIR absorption spectra resulting from increased molecular rigidity induced by boron coordination.
Kubota Y +4 more
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Gold-Catalyzed 1,3-Thiazine Formation and Uncommon Tautomer Isolation. [PDF]
J Org Chem, 2022 This work represents the first example of a gold-catalyzed formation of 1, 3-thiazine/1, 3-thiazinane by means of a catalytic approach and further uncommon isolation of the two tautomers.
Canudo-Barreras G +3 more
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