Results 21 to 30 of about 1,407 (189)
The synthesis and physico-chemical properties of new 6-acetylamino or 6-benzoyl-amino 2-benzylidene-4-methyl-4H-benzo[1,4]thiazin-3-ones and 6-benzoylamino or 6-nitro 2-benzylidene-4H-benzo[1,4]thiazin-3-ones are described.
Ana Maria Alves de Souza +6 more
doaj +3 more sources
Novel applications of the "t-amino effect" in heterocyclic chemistry. Synthesis of a pyrrolo[1,2-a]quinazoline and 5H-pyrrolo[1,2-a][3,1]benzothiazines [PDF]
1-(1-Pyrrolidinyl)benzenes substituted with an imino- or an in situ generated thiocarbonyl group in the 2-position rearrange upon heating to quinazoline and benzothiazine derivatives ...
Hamzink, M.R.J. +3 more
core +3 more sources
(R)-(−)-2-[(5-Oxido-5-phenyl-5λ4-isoquino[4,3-c][2,1]benzothiazin-12-yl)amino]benzonitrile
Copper-catalyzed cross-coupling between (S)-S-methyl-S-phenylsulfoximine (1) and 2-iodobenzonitrile (2) resulted in the discovery of an unprecedented one-pot triple arylation sequence to give (R)-(−)-2-[(5-oxido-5-phenyl-5λ4-isoquino[4,3-c][2,1 ...
Marcus Frings +2 more
doaj +1 more source
Synthesis and bioassay of azolyl benzothiazine carboxamides [PDF]
Cyclic sulfonamides (sultams) gained importance due to their potential pharmaceutical activity. Amongst these, 1,2-benzothiazine-1,1-dioxide and their derivatives represent the most familiar class of non-steroidal anti- inflammatory drugs (NSAIDs) available in the market.
Siva Sankar, P. +3 more
openaire +3 more sources
Bird Integumentary Melanins: Biosynthesis, Forms, Function and Evolution [PDF]
Melanins are the ubiquitous pigments distributed in nature. They are one of the main pigments responsible for colors in living cells. Birds are among the most diverse animals regarding melanin-based coloration, especially in the plumage, although they ...
Agrup +40 more
core +2 more sources
Synthesis of Some New 2-Methyl -1,4-benzothiazine-3(1H)- one Derivatives as Potential Vasodilators
The increase in the internal diameter of a blood vessel that results from relaxation of smooth muscle within the wall of the vessel is vasodilation. This causes an increase in blood flow and a decrease in systemic vascular resistance.
M. B. Deshmukh +2 more
doaj +1 more source
Methyl 2-(benzenesulfonamido)acetate
The title compound, C9H11NO4S, is of interest as a precursor to biologically active benzothiazines. The crystal structure is stabilized by intermolecular N—H...O and C—H...O interactions.
Muhammad Nadeem Arshad +3 more
doaj +1 more source
Synthesis of quinazolino‐1,3‐benzothiazine derivatives
AbstractThe ring‐closure reactions of N‐(3,4‐dimethoxyphenylthiomethyl)‐2‐nitrobenzamide derivatives 5a,b with phosphoryl chloride gave 4‐(2‐nitrophenyl)‐2H1,3‐benzothiazine derivatives 7a,b, which on reduction yielded 4‐(2′‐aminophenyl)‐3,4‐dihydro‐2H‐1,3‐benzothiazines 8a,b.
Szabó János +5 more
openaire +2 more sources
Synthesis and Oligonucleotide Incorporation of Fluorescent Cytosine Analogue tC: a Promising Nucleic Acid Probe [PDF]
The tricyclic cytosine, tC, is a fluorescent base analogue with excellent properties for investigating intrinsic characteristics of nucleic acid as well as interactions between nucleic acids and other molecules.
A Holmén +32 more
core +1 more source
Methyl (4-bromobenzenesulfonamido)acetate
The title compound, C9H10BrNO4S, is an intermediate for the formation of benzothiazines. In the crystal structure, intermolecular N—H...O hydrogen bonds link the molecules, forming R22(10) ring motifs, which are linked into a two-dimensional ...
Muhammad Shafiq +4 more
doaj +1 more source

