Results 51 to 60 of about 3,554 (196)

Diversity-oriented synthesis of dihydrobenzoxazepinones by coupling the Ugi multicomponent reaction with a Mitsunobu cyclization

open access: yesBeilstein Journal of Organic Chemistry, 2014
An operationally simple protocol for the synthesis of 2,3-dihydrobenzo[f][1,4]oxazepin-3-ones, based on an Ugi reaction of an ortho-(benzyloxy)benzylamine, glycolic acid, an isocyanide and an aldehyde, followed by an intramolecular Mitsunobu substitution
Lisa Moni   +4 more
doaj   +1 more source

Metal-Free Oxidative Coupling of Benzylamines to Imines under an Oxygen Atmosphere Promoted Using Salicylic Acid Derivatives as Organocatalysts

open access: yesACS Omega, 2016
The oxidative coupling of benzylamines proceeds efficiently using salicylic acid derivatives as organocatalysts under an oxygen atmosphere, affording the corresponding N-benzylidenebenzylamines in high yields.
Chun-ping Dong   +6 more
doaj   +2 more sources

Design and synthesis of 4-nitroimidazole derivatives with potential antitubercular activity

open access: yesТонкие химические технологии, 2023
Objectives. To develop the procedures for synthesis of hybrid molecules with potential anti-tubercular activity containing heterocyclic cores of 4-nitroimidazole and 1,3,4-thiadiazole within the framework of a double-drug strategy and predict bioactivity
T. S. Vedekhina   +2 more
doaj   +1 more source

Pd(II)-Catalyzed Ortho-Trifluoromethylation of Benzylamines

open access: yes, 2016
The Pd(II)-catalyzed ortho-C–H trifluoromethylation of benzylamines has been achieved utilizing an electrophilic CF3 reagent. Additives, such as H2O and Ag2O, were found to be crucial for obtaining good yields.
Jin-Quan Yu (1303500)   +3 more
core   +1 more source

Carbon Dioxide-Mediated C(sp2)–H Arylation of Primary and Secondary Benzylamines [PDF]

open access: yes, 2018
Carbon-carbon bond formation by transition metal-catalyzed C–H activation has become an important strategy to fabricate new bonds in a rapid fashion.
Mohit, Kapoor   +2 more
core   +2 more sources

Synthese von Aminocyclopropanen durch redoxneutrale Aminoalkylierung

open access: yesAngewandte Chemie, EarlyView.
Wir berichten über eine Synthese von Aminocyclopropanen durch Hydroaminoalkylierung unter Einsatz kostengünstiger, leicht zugänglicher Ausgangsmaterialien. Der Ansatz bietet Orthogonalität zu gängigen Methoden und ermöglicht eine breite Toleranz gegenüber funktionellen Gruppen.
Gwyndaf A. Oliver   +6 more
wiley   +1 more source

Expeditious Synthesis of Phenanthridines from Benzylamines via Dual Palladium Catalysis

open access: yes, 2016
A method for the synthesis of phenanthridines from benzylamines and aryl iodides which uses a dual palladium-catalyzed process is developed. The domino sequence ends via an intramolecular amination and an oxidative dehydrogenation. No protecting group or
Emmanuel Lacôte (1771780)   +6 more
core   +2 more sources

Rates of reaction of benzylamines with 1-chloro 2.4-dinitrobenzene

open access: yes, 1963
Several meta and para substituted benzylamines have been prepared. The rates of reaction of benzylamine and fourteen substituted benzylamines with 1-chloro 2,4-dinitrobenzene in ethanol have been measured. The kinetics were followed by using an acid-base
Hickford, R. S. H.
core   +1 more source

Incorporating a DAD-Type Benzothiadiazole Photosensitizer into MOFs for Photocatalytic Oxidation of Phenylsulfides and Benzylamines

open access: yes, 2023
Oxidation and removal of highly toxic sulfides and amines are particularly important for environmental and human security but remain challenging. Here, incorporating an excellent photosensitizer, donor–acceptor–donor (D–A–D)-type 4,4′-(benzo[c][1,2,5 ...
Peng-Hui Pan (13139819)   +21 more
core   +1 more source

Multicomponent reactions for DNA‐encoded library construction: Scaffold diversity and reaction engineering strategies

open access: yesBulletin of the Korean Chemical Society, EarlyView.
Abstract DNA‐encoded libraries (DELs) enable large‐scale screening for hit identification, but accessing sp3‐rich, three‐dimensional chemotypes beyond flat, aromatic scaffolds remains challenging. Multicomponent reactions (MCRs) assemble such complexity from simple building blocks in a single step, and reaction‐engineering strategies have extended on ...
Jimin Moon   +3 more
wiley   +1 more source

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