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Journal of Chemical Education, 2001
The utilization of the Biginelli reaction, a one-pot condensation of an aldehyde, a β-keto ester, and urea, is described. This reaction involves a number of individual steps, each of which is accessible to first-year organic students. The product, a 3,4-dihydropyrimidinone, is a member of a medicinally useful class of compounds.
Michael S. Holden, R. David Crouch
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The utilization of the Biginelli reaction, a one-pot condensation of an aldehyde, a β-keto ester, and urea, is described. This reaction involves a number of individual steps, each of which is accessible to first-year organic students. The product, a 3,4-dihydropyrimidinone, is a member of a medicinally useful class of compounds.
Michael S. Holden, R. David Crouch
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2‐Phenacylbenzothiazole in the Biginelli Reaction.
ChemInform, 2002AbstractFor Abstract see ChemInform Abstract in Full Text.
I. B. Dzvinchuk +2 more
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An Inexpensive Protocol for Biginelli Reaction
Synthetic Communications, 2004AbstractFor Abstract see ChemInform Abstract in Full Text.
A. Manjula +2 more
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Pietro Biginelli: The Man Behind the Reaction
European Journal of Organic Chemistry, 2011AbstractThe Biginelli dihydropyrimidine synthesis is one of the most important and oldest multicomponent reactions and has been extensively investigated in terms of application and mechanism. Surprisingly, little information is available on its discoverer, the Piedmontese chemist Pietro Biginelli, who also carried out the first studies on the ...
TRON, Gian Cesare +2 more
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Aminoheterocycles as synthons for combinatorial Biginelli reactions
Molecular Diversity, 2010Chlorotrimethylsilane (TMSCl) has been utilized as an efficient promoter and water scavenger in the synthesis of diverse dihydropyrimidines via Biginelli type MCR-heterocyclization using aminoheterocycles. High yields and a simple workup of target compounds enable the facile generation of combinatorial libraries comprising more than 2,000 compounds of ...
Sergey V, Ryabukhin +4 more
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Recent progress in asymmetric Biginelli reaction
Molecular Diversity, 2013The Biginelli reaction, which involves the interaction of ethyl acetoacetate, urea, and an appropriate aryl aldehyde, was first discovered by Pietro Biginelli about 120 years ago. The Biginelli products (3,4-dihydropyrimidin-2(1H)-ones) are interesting materials due to their significant pharmacological and structural profiles.
Majid M, Heravi +2 more
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Tandem Hydroformylation-Biginelli Reaction
Synlett, 2013The combination of a tandem process with a multicomponent reaction is a new approach to high atom-economic synthesis. A tandem hydroformylation–Biginelli reaction sequence has been developed leading to a variety of functionalized 4-alkyl-substituted 3,4-dihydropyrimidin-2(1H)-ones.
Fuchs, Daniela +4 more
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ChemInform, 2007
AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.
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AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.
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Organosilane sulfonated graphene oxide in the Biginelli and Biginelli-like reactions
New Journal of Chemistry, 2016The acid functionalized SSi-GO was used as a highly active, selective and reusable catalyst to improve the formation of pyrimidinones.
Javad Safari +2 more
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Biginelli Reaction: A Green Perspective
Current Organic Chemistry, 2012The Biginelli Reaction is a one-pot acid catalysed cyclocondensation of -keto ester, urea and aromatic aldehyde which leads to the synthesis of functionalised 3,4-dihydro-2(H)-pyrimidinones (DHPMs). This three-component reaction for the synthesis of dihydro- pyrimidinone and corresponding dihydropyrimidinethiones has now been known for more than a ...
Siva S. Panda +2 more
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