Electrophilic Trifluoromethylselenolation of Boronic Acids [PDF]
Trifluoromethylselenylated compounds are emergent compounds with interesting physicochemical properties that still suffer from a lack of efficient synthetic methods.
Clément Ghiazza +2 more
doaj +6 more sources
Electrochemical Oxidation of Aryl Boronic Acids via Fluoride Activation and Alternating Polarity Electrolysis for Aryl C–P Bond Formation [PDF]
Aryl organoboron reagents play an important role in modern organic synthesis, and interest in radical‐based coupling reactions from these precursors has grown rapidly.
Enqi Feng +5 more
doaj +2 more sources
Although boronic acids are recognized primarily for their utility as reagents in transition metal-catalyzed transformations, other applications are emerging, including their use as reaction catalysts.
Hall, Dennis G.
openaire +3 more sources
Boronic Acids and Their Derivatives in Medicinal Chemistry: Synthesis and Biological Applications
Boron containing compounds have not been widely studied in Medicinal Chemistry, mainly due to the idea that this group could confer some toxicity. Nowadays, this concept has been demystified and, especially after the discovery of the drug bortezomib, the
Mariana Pereira Silva +3 more
doaj +3 more sources
Peptide Boronic Acids by Late‐Stage Hydroboration on the Solid Phase [PDF]
Organoboron compounds have a wide range of applications in numerous research fields, and methods to incorporate them in biomolecules are much sought after.
Marius Werner +7 more
doaj +2 more sources
Alternative boronic acids in the detection of Mycolactone A/B using the thin layer chromatography (f-TLC) method for diagnosis of Buruli ulcer [PDF]
Background Mycobacterium ulcerans is the causative agent of Buruli ulcer. The pathology of M. ulcerans disease has been attributed to the secretion of a potent macrolide cytotoxin known as mycolactone which plays an important role in the virulence of the
Gideon A. Akolgo +3 more
doaj +2 more sources
Cu-Catalyzed Cross-Coupling of Nitroarenes with Aryl Boronic Acids to Construct Diarylamines. [PDF]
The development and study of a simple copper-catalyzed reaction of nitroarenes with aryl boronic acids to form diarylamines that uses phenyl silane as the stoichiometric terminal reductant is described.
Guan X, Zhu H, Driver TG.
europepmc +4 more sources
Coupling Reactions of Anhydro-Aldose Tosylhydrazones with Boronic Acids [PDF]
A catalyst-free coupling reaction between O-peracetylated, O-perbenzoylated, O-permethylated, and O-permethoxymethylated 2,6-anhydro-aldose tosylhydrazones (C-(β-d-glycopyranosyl)formaldehyde tosylhydrazones) and aromatic boronic acids is reported.
Tímea Kaszás +6 more
doaj +2 more sources
Boronic Acids as Bioorthogonal Probes for Site‐Selective Labeling of Proteins
Over the past two decades, bioorthogonal chemistry has become a preferred tool to achieve site‐selective modifications of proteins. However, there are only a handful of commonly applied bioorthogonal reactions and they display some limitations, such as ...
Dennis G Hall
exaly +2 more sources
Copper-mediated aerobic trifluoromethyltelluration of boronic acids with [Me4N][TeCF3] [PDF]
Summary: A copper-mediated trifluoromethyltelluration of arylboronic acids with [Me4N][TeCF3] using air as an environmental friendly oxidant is presented. The reaction proceeded smoothly under mild conditions in the presence of Cu(OTf)2 and bipyridine to
Jing-Yan Dong +3 more
doaj +2 more sources

