Results 101 to 110 of about 4,239 (221)

A QSAR study of a series of beta-carbolines.

, 1989
The relationship between chemical structure and biological activity of a series of beta-carbolines is studied. A chromatographic system based on Thin Layer Chromatography is used to experimentally determine lipophilicity of the investigated beta ...
G. L. Biagi, M. C. Guerra, A. M. Barbaro, BOREA, Pier Andrea, M. Recanatini, PIETROGRANDE, Maria Chiara   +5 more
core  

Oxidation of Tetrahydro-β-carbolines by Persulfate

, 2019
The development of persulfate-mediated oxidation of tetrahydro-β-carbolines is reported. This mild reaction facilitates the formation of a variety of 2-formyl N-substituted tryptamines and the related derivatives as key intermediates in moderate to ...
Haijun Chen (580445), Jing Luo (146659), Yu Gao (69071), Fu Ye (7036157), Jing Luo, Fu Ye, Haijun Chen, Yu Gao   +7 more
core   +1 more source

One-Pot Synthesis of α-Carbolines via Sequential Palladium-Catalyzed Aryl Amination and Intramolecular Arylation

, 2016
A one-pot synthesis of α-carbolines via a palladium-catalyzed aryl amination followed by intramolecular arylation is described. 2,3-Dichloro- and 2,3-dibromopyridines have been shown to react with readily available anilines to obtain various substituted ...
Philip Petrou (2379808), Joydev K. Laha (1470892), Gregory D. Cuny (249276)   +2 more
core   +1 more source

Versatile synthesis of functionalized β- and γ-carbolines via Pd-catalyzed C–H addition to nitriles/cyclization sequences

, 2018
A diverse synthesis of functionalized β-carbolines and γ-carbolines via Pd-catalyzed C–H addition of indole to nitrile/cyclization sequences is described.
Wei-Wei Liao, Ting-Ting Wang, Di Zhang
core   +1 more source

Design and Synthesis of Fluorescent 1,3-Diaryl-β-carbolines and 1,3-Diaryl-3,4-dihydro-β-carbolines

ACS Omega, 2021
JiYang Pu, Biao Chen, Wanhua Wu, Cheng Yang, Guoqing Zhang, Jason J. Chruma   +5 more
doaj   +1 more source

Catalytic enantioselective nitrone cycloadditions enabling collective syntheses of indole alkaloids

Nature Communications
Tetrahydro-β-carboline skeletons are prominent and ubiquitous in an extraordinary range of indole alkaloid natural products and pharmaceutical compounds. Powerful synthetic approaches for stereoselective synthesis of tetrahydro-β-carboline skeletons have
Xiaochen Tian, Tengfei Xuan, Jingkun Gao, Xinyu Zhang, Tao Liu, Fengbiao Luo, Ruochen Pang, Pengcheng Shao, Yun-Fang Yang, Yang Wang   +9 more
doaj   +1 more source

Pharmacological landscape of carbolines: a holistic view. [PDF]

RSC Med Chem
Zhang Y, Wu F, Rehman MU, Long S.
europepmc   +1 more source

Editorial: Psychedelic substances and neurological diseases: from basics to clinical application. [PDF]

Front Pharmacol
Linardi A, Caetano AL, Ureshino RP.
europepmc   +1 more source

Employment of Two-Acid Promoter System in Pictet-Spengler Reaction: A Robust Two-Step Synthesis of Aza-Heterocycles. [PDF]

ACS Omega
Gentili D, Lupidi G, Catalini F, Petrellini A, Ponnarassery Aravindakshan V, Rossi FV, Guzzini A, Di Giambattista G, Cimarelli C, Gabrielli S, Marcantoni E.   +10 more
europepmc   +1 more source

β-Carboline: a privileged scaffold from nature for potential antimalarial activity. [PDF]

RSC Med Chem
Punmiya A, Pandey AR, Vora A.
europepmc   +1 more source