Results 131 to 140 of about 1,477,235 (156)

Signal Propagation in the ATPase Domain of <i>Mycobacterium tuberculosis</i> DNA Gyrase from Dynamical-Nonequilibrium Molecular Dynamics Simulations. [PDF]

Biochemistry
Kamsri B, Kamsri P, Punkvang A, Chimprasit A, Saparpakorn P, Hannongbua S, Spencer J, Oliveira ASF, Mulholland AJ, Pungpo P.   +9 more
europepmc   +1 more source

Two classes of DNA gyrase inhibitors elicit distinct evolutionary trajectories toward resistance in gram-negative pathogens. [PDF]

NPJ Antimicrob Resist
Leyn SA, Kent JE, Zlamal JE, Elane ML, Vercruysse M, Osterman AL.   +5 more
europepmc   +1 more source

New N-amino-5-cyano-6-pyridones as antimicrobial small molecules endowed with DNA gyrase a inhibitory activity: design, one-pot synthesis, biological assessment and in silico insights. [PDF]

BMC Chem
Kamaly OA, Younes AS, Harras MF, Sabour R, Alsfouk AA, Ibrahim MH.   +5 more
europepmc   +1 more source

Ligand-Based Virtual Screening for Discovery of Indole Derivatives as Potent DNA Gyrase ATPase Inhibitors Active against Mycobacterium tuberculosis and Hit Validation by Biological Assays. [PDF]

J Chem Inf Model
Pakamwong B, Thongdee P, Kamsri B, Phusi N, Taveepanich S, Chayajarus K, Kamsri P, Punkvang A, Hannongbua S, Sangswan J, Suttisintong K, Sureram S, Kittakoop P, Hongmanee P, Santanirand P, Leanpolchareanchai J, Spencer J, Mulholland AJ, Pungpo P.   +18 more
europepmc   +1 more source

Dynamic Profiling and Binding Affinity Prediction of NBTI Antibacterials against DNA Gyrase Enzyme by Multidimensional Machine Learning and Molecular Dynamics Simulations. [PDF]

ACS Omega
Kokot M, Minovski N.
europepmc   +1 more source

Multimodal antibacterial potency of newly designed and synthesized Schiff's/Mannich based coumarin derivatives: potential inhibitors of bacterial DNA gyrase and biofilm production. [PDF]

RSC Adv
Pakeeraiah K, Swain PP, Sahoo A, Panda PK, Mahapatra M, Mal S, Sahoo RK, Sahu PK, Paidesetty SK.   +8 more
europepmc   +1 more source

Structure of Escherichia coli DNA gyrase with chirally wrapped DNA supports ratchet-and-pawl mechanism for an ATP-powered supercoiling motor

Michalczyk E, Pabiś M, Heddle J, Ghilarov D.   +3 more
europepmc   +1 more source

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Novel and Structurally Diversified Bacterial DNA Gyrase Inhibitors Discovered through a Fluorescence-Based High-Throughput Screening Assay

ACS Pharmacology and Translational Science, 2022
Prem P Chapagain, Jeremy W. Chambers, Fenfei Leng   +2 more
exaly  

Recent advances in DNA gyrase-targeted antimicrobial agents

European Journal of Medicinal Chemistry, 2020
Trudi Collet, Satish N Dighe
exaly  

DNA Gyrase: Structure and Function

Critical Reviews in Biochemistry and Molecular Biology, 1991
Anthony Maxwell
exaly