Results 121 to 130 of about 1,477,235 (156)

Structural basis of chiral wrap and T-segment capture by <i>Escherichia coli</i> DNA gyrase. [PDF]

Proc Natl Acad Sci U S A
Michalczyk E, Pakosz-Stępień Z, Liston JD, Gittins O, Pabis M, Heddle JG, Ghilarov D.   +6 more
europepmc   +1 more source

Computational identification of novel natural inhibitors against triple mutant DNA gyrase A in fluoroquinolone-resistant Salmonella Typhimurium. [PDF]

Biochem Biophys Rep
Haryini S, Doss C GP.
europepmc   +1 more source

Microbial-based natural products as potential inhibitors targeting DNA gyrase B of Mycobacterium tuberculosis: an in silico study. [PDF]

Front Chem
Elsaman T, Mohamed MA, Mohamed MS, Eltayib EM, Abdalla AE.   +4 more
europepmc   +1 more source

Macrolones target bacterial ribosomes and DNA gyrase and can evade resistance mechanisms. [PDF]

Nat Chem Biol
Aleksandrova EV, Ma CX, Klepacki D, Alizadeh F, Vázquez-Laslop N, Liang JH, Polikanov YS, Mankin AS.   +7 more
europepmc   +1 more source

In Silico Study of the Potential Inhibitory Effects on Escherichia coli DNA Gyrase of Some Hypothetical Fluoroquinolone-Tetracycline Hybrids. [PDF]

Pharmaceuticals (Basel)
Lungu IA, Oancea OL, Rusu A.
europepmc   +1 more source

New Benzofuran-Pyrazole-Based Compounds as Promising Antimicrobial Agents: Design, Synthesis, DNA Gyrase B Inhibition, and In Silico Studies. [PDF]

Pharmaceuticals (Basel)
Abd El-Karim SS, Anwar MM, Syam YM, Awad HM, El-Dein AN, El-Ashrey MK, Alkahtani HM, Abdelwahed SH.   +7 more
europepmc   +1 more source

Structural basis of DNA crossover capture by <i>Escherichia coli</i> DNA gyrase. [PDF]

Science
Vayssières M, Marechal N, Yun L, Lopez Duran B, Murugasamy NK, Fogg JM, Zechiedrich L, Nadal M, Lamour V.   +8 more
europepmc   +1 more source

Synthesis and Antimicrobial Evaluation of New 1,2,4-Triazolo[1,5-a]pyrimidine-Based Derivatives as Dual Inhibitors of Bacterial DNA Gyrase and DHFR. [PDF]

ACS Omega
Al-Wahaibi LH, Rabea SM, Mahmoud MA, Youssif BGM, Bräse S, Abdel-Aziz SA.   +5 more
europepmc   +1 more source

New N-phenylpyrrolamide inhibitors of DNA gyrase with improved antibacterial activity. [PDF]

RSC Adv
Cotman AE, Fulgheri F, Piga M, Peršolja P, Tiz DB, Skok Ž, Durcik M, Sterle M, Dernovšek J, Cruz CD, Tammela P, Szili PÉ, Daruka L, Pál C, Zega A, Mašič LP, Ilaš J, Tomašič T, Kikelj D, Zidar N.   +19 more
europepmc   +1 more source

Identification of Anti-Tuberculosis Drugs Targeting DNA Gyrase A and Serine/Threonine Protein Kinase PknB: A Machine Learning-Assisted Drug-Repurposing Approach. [PDF]

Trop Med Infect Dis
Lee D, Islam MA, Natarajan S, Dudekula DB, Chung H, Park J, Oh B.   +6 more
europepmc   +1 more source