Results 101 to 110 of about 19,626 (172)

Spiropyrimidinetrione DNA Gyrase Inhibitors with Potent and Selective Antituberculosis Activity. [PDF]

J Med Chem, 2022
Govender P, Müller R, Singh K, Reddy V, Eyermann CJ, Fienberg S, Ghorpade SR, Koekemoer L, Myrick A, Schnappinger D, Engelhart C, Meshanni J, Byl JAW, Osheroff N, Singh V, Chibale K, Chibale K, Basarab GS.   +17 more
europepmc   +1 more source

Phytochemical profiling of Vitex negundo seeds via UHPLC-QTOF-MS/MS analyses with antimicrobial evaluation and in silico targeting of DNA Gyrase B and Secreted Aspartic Proteinase 2 (SAP2). [PDF]

PLoS One
Mustafa J, Ashraf T, Ali B, Kousar S, Mahmood A, Ullah S, Imran M, Ali B, Rahim U, Yunis M.   +9 more
europepmc   +1 more source

An In-Silico Evaluation of Anthraquinones as Potential Inhibitors of DNA Gyrase B of Mycobacterium tuberculosis. [PDF]

Microorganisms, 2022
Amorim JC, Cabrera Bermeo AE, Vásquez Urgilés VE, Martínez León MR, Carpio Arévalo JM.   +4 more
europepmc   +1 more source

In vitro and in silico evaluation of phytocompounds from Leucaena leucocephala and Entada phaseoloides targeting DNA gyrase, topoisomerase II, AKT1. [PDF]

Sci Rep
Khiangte L, Sailo H, Ralte L, Lalnunmawia F, Senthilkumar N, Singh YT.   +5 more
europepmc   +1 more source

Isoflavonoid and Furanochromone Natural Products as Potential DNA Gyrase Inhibitors: Computational, Spectral, and Antimycobacterial Studies. [PDF]

ACS Omega, 2023
Jagatap VR, Ahmad I, Sriram D, Kumari J, Adu DK, Ike BW, Ghai M, Ansari SA, Ansari IA, Wetchoua POM, Karpoormath R, Karpoormath R, Patel H.   +12 more
europepmc   +1 more source

Structural basis of chiral wrap and T-segment capture by Escherichia coli DNA gyrase. [PDF]

Proc Natl Acad Sci U S A
Michalczyk E, Pakosz-Stępień Z, Liston JD, Gittins O, Pabis M, Heddle JG, Ghilarov D.   +6 more
europepmc   +1 more source

Structural Aspects of Mycobacterium tuberculosis DNA Gyrase Targeted by Novel Bacterial Topoisomerase Inhibitors. [PDF]

ACS Med Chem Lett
Kokot M, Hrast Rambaher M, Feng L, Mitchenall LA, Lawson DM, Maxwell A, Parish T, Minovski N, Anderluh M.   +8 more
europepmc   +1 more source

Computational identification of novel natural inhibitors against triple mutant DNA gyrase A in fluoroquinolone-resistant Salmonella Typhimurium. [PDF]

Biochem Biophys Rep
Haryini S, Doss C GP.
europepmc   +1 more source

Microbial-based natural products as potential inhibitors targeting DNA gyrase B of Mycobacterium tuberculosis: an in silico study. [PDF]

Front Chem
Elsaman T, Mohamed MA, Mohamed MS, Eltayib EM, Abdalla AE.   +4 more
europepmc   +1 more source

In Silico Study of the Potential Inhibitory Effects on Escherichia coli DNA Gyrase of Some Hypothetical Fluoroquinolone-Tetracycline Hybrids. [PDF]

Pharmaceuticals (Basel)
Lungu IA, Oancea OL, Rusu A.
europepmc   +1 more source