Results 11 to 20 of about 674 (175)
ChemInform Abstract: Electrochemical Oxidation of Ergolines.
ChemInform, 1992 AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable via the “References” option.
K. SEIFERT +2 more
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Ropinirole, a Non‐Ergoline Dopamine Agonist [PDF]
CNS Drug Reviews, 2005 ABSTRACTDopamine agonists have become indispensable in the treatment of Parkinson's disease. In every‐day practice, however, the decision to select the best compound for an individual patient is rendered difficult because of the large number of substances available on the market.
Wolfgang H, Jost, Dieter, Angersbach
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Pleuropulmonary changes induced by ergoline drugs [PDF]
European Respiratory Journal, 1996 Classic ergolines, such as bromocriptine, methysergide and ergotamine, can induce chronic pleuropneumonitis. We present the cases of eight patients who developed similar changes whilst on other ergolines. In this retrospective case study spanning 1985-1995, clinical data, radiological material, pulmonary function, bronchoalveolar lavage and ...
P, Pfitzenmeyer +7 more
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Two new dopamine agonists that are long acting in vivo but short acting in vitro.
, 1980 The effects of two new ergolines, pergolide and CH29-717, on prolactin secretion in vitro and in vivo were compared with those of bromocriptine. Both ergolines had in vitro potencies similar to that of bromocriptine, but had a shorter duration of action.
Grossman, Ashley +5 more
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Stimulant and hallucinogenic novel psychoactive substances; an update [PDF]
, 2023 Introduction: The renewed interest in considering a range of stimulants, psychedelics and dissociatives as therapeutics emphasizes the need to draft an updated overview of these drugs’ clinical and pharmacological issues.
Amira Guirguis
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Special ergolines efficiently inhibit the chemokine receptor CXCR3 in blood
, 2011 The structure activity relationship of highly potent special ergolines which selectively block the chemokine receptor CXCR3 is reported. The most potent compounds showed IC50 values below 10 nM in both ligand binding and Ca2+-mobilization assays. However,
Baenteli, Rolf +6 more
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, 2014 Ergolines were recently identified as a novel class of H3-Receptor (H3R) inverse agonist. While their optimization led to drug candidates with encouraging properties for the treatment of narcolepsy, brain penetration remained low. To overcome this issue,
Zhang, Xuechun +13 more
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Electrochemical synthesis of 2-haloergolines
, 1987 Regiosclective halogenation (chlorination, bromination, iodination) of several ergolines to the corresponding 2-halo derivatives was performed in moderate to good yields by potential controlled electrolysis at platinum in acetonitrile in the presence of ...
G. FIORI +3 more
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Genetics of ergoline alkaloid formation in Penicillium roquefortii [PDF]
Applied and Environmental Microbiology, 1985 Auxotrophic, spore color, and alkaloid biosynthetic mutants of Penicillium roquefortii were selected after N-methyl-N'-nitro-N-nitrosoguanidine treatment. Diploids were obtained via protoplast fusion techniques, and the segregants from a diploid were genetically analyzed. The data demonstrated the potential of parasexual recombination in this organism.
S L, Hong, J E, Robbers
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Respirology, EarlyView.We tested the respective effect of high‐flow and supplemental O2 from nasal high‐flow O2 therapy (NHFO2) on dyspnea and exercise tolerance in fibrotic interstitial lung disease. Supplemental O2 and NHFO2 (but not high‐flow) provided improvements in these outcomes at “iso‐O2 saturation” due to reduced ventilatory requirements.
Sarah Thivent +4 more
wiley +1 more source