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Az irreverzibilis antagonista FSCPX hatása az A1 adenozin receptor-mediálta direkt negatív inotrópiára patkány és tengerimalac bal pitvaron a SABRE modellel meghatározva

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The Surmountable Effect of FSCPX, an Irreversible A1 Adenosine Receptor Antagonist, on the Negative Inotropic Action of A1 Adenosine Receptor Full Agonists in Isolated Guinea Pig Left Atria

Archives of Pharmacal Research, 2013
A1 adenosine receptors (A1 receptors) are widely expressed in mammalian tissues; therefore attaining proper tissue selectivity is a cornerstone of drug development. The fact that partial agonists chiefly act on tissues with great receptor reserve can be exploited to achieve an appropriate degree of tissue selectivity.
Rudolf Gesztelyi, Judit Zsuga, Mariann Bombicz   +2 more
exaly   +3 more sources

A Body of Circumstantial Evidence for the Irreversible Ectonucleotidase Inhibitory Action of FSCPX, an Agent Known as a Selective Irreversible A1 Adenosine Receptor Antagonist so Far

International Journal of Molecular Sciences, 2021
Rudolf Gesztelyi, Béla Juhász, Judit Zsuga   +2 more
exaly  

An Advanced in Silico Modelling of the Interaction Between FSCPX, an Irreversible A1 Adenosine Receptor Antagonist, and NBTI, a Nucleoside Transport Inhibitor, in the Guinea Pig Atrium

Molecules, 2019
Rudolf Gesztelyi, Béla Juhász, Ákos Pintér   +2 more
exaly  

Synthesis and Use of FSCPX, an Irreversible Adenosine A1 Antagonist, as a ‘Receptor Knock-Down’ Tool

Bioorganic and Medicinal Chemistry Letters, 2001
Adriaan P IJzerman, Piet H van der Graaf, Jacqueline E van Muijlwijk-Koezen   +2 more
exaly  

New Irreversible Adenosine A1 Antagonists Based on FSCPX

Bioorganic and Medicinal Chemistry Letters, 2002
Peter J. Scammells, Stephen P Baker
exaly  

Differential A1 Adenosine Receptor Reserve for Two Actions of Adenosine on Guinea Pig Atrial Myocytes

Molecular Pharmacology, 1997
Stephen P Baker, John C Shryock, Donn M Dennis   +2 more
exaly  

A Novel Irreversible Antagonist of the A1-Adenosine Receptor.

Molecular Pharmacology, 1996
Peter J. Scammells, Stephen P Baker, L Belardinelli   +2 more
exaly  

Fluorosulfonyl-Substituted Xanthines as Selective Irreversible Antagonists for the A1-Adenosine Receptor

Journal of Medicinal Chemistry, 2000
Peter J. Scammells, Stephen P Baker
exaly  

Modulation of Agonist Responses at the A1 Adenosine Receptor by an Irreversible Antagonist, Receptor–G Protein Uncoupling and by the G Protein Activation State

Biochemical Pharmacology, 2002
Adriaan P IJzerman, Anna Lorenzen, Heidrun Lang   +2 more
exaly