Results 31 to 40 of about 85 (60)

The ability of SABRE, a new quantitative receptor function model, to quantify receptor binding from even challenging concentration-effect data with a single unified fit. [PDF]

Front Pharmacol
Olah B, Tarjanyi V, Viczjan G, Ovari I, Csoto A, Szilvassy Z, Juhasz B, Zsuga J, Gesztelyi R, Erdei T.   +9 more
europepmc   +1 more source

A Non-imaging High Throughput Approach to Chemical Library Screening at the Unmodified Adenosine-A₃ Receptor in Living Cells. [PDF]

Front Pharmacol, 2017
Arruda MA, Stoddart LA, Gherbi K, Briddon SJ, Kellam B, Hill SJ.   +5 more
europepmc   +1 more source

The flexibility of SABRE, a new quantitative receptor function model, when fitting challenging concentration-effect data. [PDF]

Front Pharmacol
Olah B, Tarjanyi V, Takacs B, Pluzsnyik E, Viczjan G, Ovari I, Szilvassy Z, Juhasz B, Zsuga J, Erdei T, Gesztelyi R.   +10 more
europepmc   +1 more source

Commentary: The flexibility of SABRE, a new quantitative receptor function model, in fitting challenging concentration-effect data. [PDF]

Front Pharmacol
Buchwald P.
europepmc   +1 more source

Control of enteric neuromuscular functions by purinergic A(3) receptors in normal rat distal colon and experimental bowel inflammation. [PDF]

Br J Pharmacol, 2010
Antonioli L, Fornai M, Colucci R, Ghisu N, Tuccori M, Awwad O, Bin A, Zoppellaro C, Castagliuolo I, Gaion RM, Giron MC, Blandizzi C.   +11 more
europepmc   +1 more source

Az FSCPX (irreverzibilis A1 adenozin receptor antagonista) hatását befolyásoló kinetikai sajátosságok ex vivo kísérleti körülmények között

, 2021
Takács Tímea
core  

Small Molecule, NSC95397, Inhibits the CtBP1-Protein Partner Interaction and CtBP1-Mediated Transcriptional Repression. [PDF]

J Biomol Screen, 2015
Blevins MA, Kouznetsova J, Krueger AB, King R, Griner LM, Hu X, Southall N, Marugan JJ, Zhang Q, Ferrer M, Zhao R.   +10 more
europepmc   +1 more source

Advancing Covalent Ligand and Drug Discovery beyond Cysteine. [PDF]

Chem Rev
Kim G, Grams RJ, Hsu KL.
europepmc   +1 more source

A covalent antagonist for the human adenosine A_2A receptor. [PDF]

Purinergic Signal, 2017
Yang X, Dong G, Michiels TJM, Lenselink EB, Heitman L, Louvel J, IJzerman AP.   +6 more
europepmc   +1 more source

A cell-based PDE4 assay in 1536-well plate format for high-throughput screening. [PDF]

J Biomol Screen, 2008
Titus SA, Li X, Southall N, Lu J, Inglese J, Brasch M, Austin CP, Zheng W.   +7 more
europepmc   +1 more source