Results 41 to 50 of about 85 (60)

Inhibitors of the apurinic/apyrimidinic endonuclease 1 (APE1)/nucleophosmin (NPM1) interaction that display anti-tumor properties. [PDF]

Mol Carcinog, 2016
Poletto M, Malfatti MC, Dorjsuren D, Scognamiglio PL, Marasco D, Vascotto C, Jadhav A, Maloney DJ, Wilson DM, Simeonov A, Tell G.   +10 more
europepmc   +1 more source

Covalent Allosteric Probe for the Metabotropic Glutamate Receptor 2: Design, Synthesis, and Pharmacological Characterization. [PDF]

J Med Chem, 2019
Doornbos MLJ, Wang X, Vermond SC, Peeters L, Pérez-Benito L, Trabanco AA, Lavreysen H, Cid JM, Heitman LH, Tresadern G, IJzerman AP.   +10 more
europepmc   +1 more source

Purinergic receptors and gastrointestinal secretomotor function. [PDF]

Purinergic Signal, 2008
Christofi FL.
europepmc   +1 more source

The identification of inhibitors of Schistosoma mansoni miracidial transformation by incorporating a medium-throughput small-molecule screen. [PDF]

Exp Parasitol, 2010
Taft AS, Norante FA, Yoshino TP.
europepmc   +1 more source

The influence of the way of regression on the results obtained by the receptorial responsiveness method (RRM), a procedure to estimate a change in the concentration of a pharmacological agonist near the receptor. [PDF]

Front Pharmacol
Ovari I, Viczjan G, Erdei T, Takacs B, Tarjanyi V, Zsuga J, Szucs M, Szilvassy Z, Juhasz B, Gesztelyi R.   +9 more
europepmc   +1 more source

An Affinity-Based Probe for the Human Adenosine A_2A Receptor. [PDF]

J Med Chem, 2018
Yang X, Michiels TJM, de Jong C, Soethoudt M, Dekker N, Gordon E, van der Stelt M, Heitman LH, van der Es D, IJzerman AP.   +9 more
europepmc   +1 more source

Design and pharmacological characterization of VUF14480, a covalent partial agonist that interacts with cysteine 98(3.36) of the human histamine H₄ receptor. [PDF]

Br J Pharmacol, 2013
Nijmeijer S, Engelhardt H, Schultes S, van de Stolpe AC, Lusink V, de Graaf C, Wijtmans M, Haaksma EE, de Esch IJ, Stachurski K, Vischer HF, Leurs R.   +11 more
europepmc   +1 more source

A comparison of an A1 adenosine receptor agonist (CVT-510) with diltiazem for slowing of AV nodal conduction in guinea-pig. [PDF]

Br J Pharmacol, 1999
Snowdy S, Liang HX, Blackburn B, Lum R, Nelson M, Wang L, Pfister J, Sharma BP, Wolff A, Belardinelli L.   +9 more
europepmc   +1 more source

Adenosine receptors and asthma. [PDF]

Handb Exp Pharmacol, 2009
Wilson CN, Nadeem A, Spina D, Brown R, Page CP, Mustafa SJ.   +5 more
europepmc   +1 more source

The surmountable effect of FSCPX, an irreversible A1 adenosine receptor antagonist, on the negative inotropic action of A1 adenosine receptor full agonists in isolated guinea pig left atria

, 2012
Pák, Krisztián
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