Results 151 to 160 of about 9,380 (213)

Distinct Phosphorylation Patterns of AT1R by Biased Ligands and GRK Subtypes. [PDF]

Int J Mol Sci
Zhang Z, Liu C, Gong J, Su C, Liu Z, Li J, Zhang H.   +6 more
europepmc   +1 more source

Signaling Bias as a Framework for Therapeutically Relevant Orthosteric Agonists: The β₂ Adrenergic Receptor Paradigm. [PDF]

Biochemistry
Georgiou K, Kolocouris A.
europepmc   +1 more source

Age-dependent impairment of dopamine D1 receptor signalling in mouse striatum by <i>FMR1</i> variant P626L. [PDF]

Brain Commun
Fu J, Jiang W, Shen L, Fu J, Duan X, Liu D, Long J, Ye S, Tang L, Yi YH, Long YS.   +10 more
europepmc   +1 more source

Development of a GRK2-inhibitory peptide

, 2017
openaire   +2 more sources

The GRK2/AP-1 Signaling Axis Mediates Vascular Endothelial Dysfunction and Atherosclerosis Induced by Oscillatory Low Shear Stress. [PDF]

Adv Sci (Weinh)
Wu LD, Shi Y, Kong CH, Chen AQ, Kang Y, Kan JY, Jiang XM, Chu P, Wang DC, Lv YF, Qian ZY, Jiang ZH, Chen YW, Sun Y, Chang RR, Zhou WY, Gu Y, Zhang JX, Chen SL.   +18 more
europepmc   +1 more source

Drug Repositioning in Doxorubicin-Induced Cardiotoxicity Protection. [PDF]

Int J Mol Sci
Kosić M, Pajović V, Jovanović M, Japundžić-Žigon N.   +3 more
europepmc   +1 more source

Efficacy of Paroxetine as an Adjuvant Therapy in Rheumatoid Arthritis Patients: A Randomized Controlled Study. [PDF]

Drug Des Devel Ther
Aldossary KM, Abdallah MS, Mosalam EM, Kamal N, Saif DS, Elsayed SA, Afifi N, Zakaraia HG, Khrieba MO, Bahaa MM.   +9 more
europepmc   +1 more source

GPCR kinases phosphorylate GPCR C-terminal peptides in a hierarchical manner. [PDF]

Commun Biol
Löbbert A, Lorz N, Matthees ESF, Rößler P, Hoffmann C, Gossert AD.   +5 more
europepmc   +1 more source

Helix-bundle and C-terminal GPCR domains differentially influence GRK-specific functions and β-arrestin-mediated regulation. [PDF]

Nat Commun
Matthees ESF, Haider RS, Klement L, Reichel M, Blum NK, Weitzel V, Trüpschuch T, Ziegler C, Drube J, Schulz S, Hoffmann C.   +10 more
europepmc   +1 more source

P-Rex1 limits the agonist-induced internalization of GPCRs independently of its Rac-GEF activity.

Cell Rep
Baker MJ, Hampson E, Islam P, Moral RP, Maunders EA, Hornigold K, Tsonou E, Malliri A, Hornigold DC, Hubbard RE, Massey AJ, Welch HCE.   +11 more
europepmc   +1 more source