Antibiotic resistance, particularly against fluoroquinolones and macrolides, has emerged globally among thermophilic Campylobacters (Campylobacter jejuni and Campylobacter coli), giving rise to concerns about the efficacy of antibiotic treatment of these
Claudia B. Barroso +4 more
doaj +1 more source
Isatin: identity with the purified endogenous monoamine oxidase inhibitor tribulin
Purified tribulin, an endogenous monoamine oxidase (MAO) inhibitor, has been identified by direct probe insertion mass spectrometry as the indole-2,3-dione, isatin.
Watkins, P.J. +5 more
core +1 more source
Counter-Current Chromatography Separation of Isatin Derivatives using the Sandmeyer Methodology
A rapid and efficient method, using high-speed counter-current chromatography (HSCCC) technique, was developed for the separation of isomeric isatin derivatives, prepared following the Sandmeyer route.
Silva, Bárbara V. +4 more
core
Early pharmacological profiling of isatin derivatives as potent and selective cytotoxic agents [PDF]
Isatin derivatives have attracted a lot of interest for their potential in the development of new anticancer drugs. A library of 38 isatin derivatives, created through an Ugi four-component reaction, underwent an initial screening in a panel of six human
Fernandes, Miguel Xavier, +16 more
core +1 more source
Design, Synthesis of New 1,2,4-Triazole/1,3,4-Thiadiazole with Spiroindoline, Imidazo[4,5-b]quinoxaline and Thieno[2,3-d]pyrimidine from Isatin Derivatives as Anticancer Agents. [PDF]
Abu-Hashem AA, Al-Hussain SA.
europepmc +1 more source
Bis-isatin derivatives: design, synthesis, and biological activity evaluation as potent dimeric DJ-1 inhibitors. [PDF]
Chen XB +9 more
europepmc +1 more source
Efficient cyclopropanation of α,β-unsaturated ketones using α-ketoesters or isatin derivatives is reported. The cyclopropanation reaction occurs via a cascade transformation that starts with addition of deprotonated dialkyl phosphite to the keto groups ...
Hui Liu (33624) +3 more
core +1 more source
Synthesis and Antiproliferatory Activities Evaluation of Multi-Substituted Isatin Derivatives. [PDF]
Ding Y +7 more
europepmc +1 more source
Novel <i>N</i>-Substituted Amino Acid Hydrazone-Isatin Derivatives: Synthesis, Antioxidant Activity, and Anticancer Activity in 2D and 3D Models <i>In Vitro</i>. [PDF]
Tumosienė I +4 more
europepmc +1 more source
Electrolytic Reduction of Isatin and Its Derivatives. I. Reduction of Isatin [PDF]
openaire +1 more source

