Results 111 to 120 of about 7,252 (218)

Synthesis, Characterization, Molecular Docking, and Antimicrobial Evaluation of New Acetylenic Mannich Bases of Isatin–Thiazole Derivatives

Iraqi Journal of Pharmaceutical Sciences
The isatin molecule is present in many natural substances, like plants and animals, and it is utilized to prepare compounds with various biological activities.
marwa hashim almusawi, May Mohammed Jawad Al-Mudhafar   +1 more
doaj   +1 more source

Isatin derivatives as broad-spectrum antiviral agents: the current landscape. [PDF]

Med Chem Res, 2022
Elsaman T, Mohamed MS, Eltayib EM, Abdel-Aziz HA, Abdalla AE, Munir MU, Mohamed MA.   +6 more
europepmc   +1 more source

Insighting isatin derivatives as potential antiviral agents against NSP3 of COVID-19. [PDF]

Chem Zvesti, 2022
Ilyas M, Muhammad S, Iqbal J, Amin S, Al-Sehemi AG, Algarni H, Alarfaji SS, Alshahrani MY, Ayub K.   +8 more
europepmc   +1 more source

Design, synthesis and anticonvulsant activity of some new 6,8-halo-substituted-2H-[1,2,4]triazino[5,6-b]indole-3(5H)-one/-thione and 6,8-halo-substituted 5-methyl-2H-[1,2,4]triazino[5,6-b]indol-3(5H)-one/-thione [PDF]

, 2014
A new series of 6,8-halo-substituted-2H-[1,2,4]triazino[5,6-b]indole-3(5H)-one/-thione and 6,8-halo-substituted 5-methyl-2H-[1,2,4]triazino[5,6-b]indol-3(5H)-one/-thione (5a-5l) were designed and synthesized keeping in view of the structural ...
Jain, Sandeep, Kumar, Rajeev, Roy, R. K., Singh, Hariram, Singh, Tejendra   +4 more
core  

Identification of novel 1,2,3-triazole isatin derivatives as potent SARS-CoV-2 3CLpro inhibitors via click-chemistry-based rapid screening. [PDF]

RSC Med Chem, 2023
Jiang X, Li J, Viayna A, Luque FJ, Woodson M, Jing L, Gao S, Zhao F, Xie M, Toth K, Tavis J, Tollefson AE, Liu X, Zhan P.   +13 more
europepmc   +1 more source

Effective heterogeneous electro-Fenton process for the degradation of a malodorous compound, indole using iron loaded alginate beads as a reusable catalyst

, 2016
International audienceIn this work the characterization and the performance of iron immobilized in alginate beads (Fe-ABs) as catalyst for heterogeneous electro-Fenton (EF) treatment of a malodorous compound, indole, was investigated.
Adhoum, Nafâa, Amrane, Abdeltif, Assadi, Aymen, Fourcade, Florence, Hammouda, Samia Ben, Monser, Lotfi, Soutrel, Isabelle   +6 more
core   +3 more sources

Cytotoxic Effects of Dibromoisatin Derivatives on Hela and HepG2 Cell Lines Using MTT Assay

Journal of Mazandaran University of Medical Sciences, 2017
Background and purpose: Tumors are one of the most important threats to human life and improving the drugs used in their treatment is always necessary.  Isatin is found in many plants and also synthesized through different methods.
Mohammad Shokrzadeh, Saied Emami, Melika Amirzadeh, Mona Modanloo   +3 more
doaj  

Evaluation of the Antibacterial Activity of Isatin against Campylobacter jejuni and Campylobacter coli Strains

Applied Microbiology
Antibiotic resistance, particularly against fluoroquinolones and macrolides, has emerged globally among thermophilic Campylobacters (Campylobacter jejuni and Campylobacter coli), giving rise to concerns about the efficacy of antibiotic treatment of these
Claudia B. Barroso, Liliane M. Seki, Wagner T. C. Esteves, Michele C. Nascimento, Aurea Echevarria   +4 more
doaj   +1 more source

Investigation of potential anti-radiation and anti-neoplastic compounds related to plant growth regulators second quarterly progress report, 1 oct. 1964 - 1 jan. 1965 [PDF]

Antiradiation and antineoplastic compounds related to plant growth regulators - cytotoxic effects and radiation ...
Norman, D., Schultz, R. D.
core   +1 more source

Synthesis kinases inhibitory potencies and in vitro antiproliferative activity of isoindigo and 7'-azaisoindigo derivatives substituted by Sonogashira cross-coupling [PDF]

, 2009
International audienceIn the course of structure–activity relationship studies we were interested in the synthesis of isoindigo and 7′-azaisoindigo derivatives substituted at the N-1 position by a 1-(2,3,4,6-tetra-O-acetyl-β-d-glucopyranosyl), at the 5 ...
Anizon, Fabrice, Bouchikhi, Fadoua, Moreau, Pascale   +2 more
core