Results 111 to 120 of about 1,834 (212)

Isoxazolines: an insight to their synthesis and diverse applications

, 2015
The five membered heterocycles isoxazolines are considered as important class of compounds in bioorganic and medicinal chemistry. They were treated as useful intermediates for transforming to large number of bioactive molecules.
Vasanth, G., Renuka, N., Ajay Kumar, K., Govindaraju, M.   +3 more
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trans-Hydroxylation of cyclopent-5-ene[d]isoxazolines

, 2020
The title reaction has been studied as a variant of the cyclopentane ring functionalization of cyclopent-5-ene[d]isoxazolines as the key intermediates in total synthesis of azaand oxo prostaglandin analogues by nitrileoxides approach.
Antonevich, I. P., Nesterova, S. V.
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Monographie sur les isoxazolines : une nouvelle famille de molécules à activité antiparasitaire externe utilisées chez les carnivores domestiques

, 2017
Ectoparasiticides targeting fleas and ticks are frequently used in domestic carnivores. The currently available drugs belong to several chemical families and most of them interfere with the nervous system of arthropods.
Lesieur, Floriane
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Effect of beta-cyclodextrin on the extraction of isoxazolines from aqueous ethanol into chloroform

, 2015
Regioisomeric pairs of isoxazolines were prepared through reaction of nitrile oxides with ethyl trans-cinnamate. The effect of β -cyclodextrin on the solubility of these compounds in aqueous ethanol and their extraction into chloroform has been ...
Lincoln, Stephen F, Vuckovic, George, Hughes, Colin, Simpson, Gregory Wayne, Easton, Christopher   +4 more
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Synthesis of novel bis heterocycles: Bis pyrroles, pyrrolyl pyrazolines and pyrrolyl isoxazolines

, 2008
1707-1712The Michael acceptors, 1-arylsulfonyl-2-styrylsulfonylethenes have been used as synthons to develop bis pyrroles, pyrrolyl pyrazolines and pyrrolyl isoxazolines by 1,3-dipolar cycloaddition of tosylmethyl isocyanide, nitrile imines and nitrile ...
Padmavathi, V, Radhalakshmi, T, Mahesh, K, Mohan, A V Nagendra   +3 more
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Discovery of mCMV280: An Oral Ectoparasiticide in the Isoxazoline Class with Reduced Mammalian Brain Exposure. [PDF]

J Med Chem
McComic SE, Wilson KB, Li Z, Chen J, Weiss F, Song L, Mazumdar W, Dvorak CA, Brittain J, Lee KJ, Li S, Joseph SB, McNamara CW, Vos MW, Sheshachalam A, Inácio A, Dechering KJ, Chatterjee AK, Swale DR.   +18 more
europepmc   +1 more source

Synthesis of mono- and di-(<i>C</i>-glycopyranosyl-isoxazol(in)yl) derivatives on aromatic scaffolds and their evaluation as anti-adherence agents of <i>Candida albicans</i>. [PDF]

Front Chem
Kaszás T, Szakács B, Blága T, Doherty K, Keenan-Dillon R, Reynolds S, Kavanagh K, Velasco-Torrijos T, Somsák L, Tóth M.   +9 more
europepmc   +1 more source

Evaluation of efficacy and pharmacokinetics of novel fluralaner tablet formulation (WellPet™) in dogs. [PDF]

Front Vet Sci
Cruz BC, Teixeira MB, de Melo Cruz GA, da Silva JADCEM, Michels MG, Pistoni CDN, Buso MAM, de Almeida FN, Gatto IRH.   +8 more
europepmc   +1 more source

Copper(II)-Photocatalyzed Radical Anellation of Nitroalkanes with Alkenes or Alkynes for the Synthesis of Isoxazolines and Isoxazoles. [PDF]

Angew Chem Int Ed Engl
Sardana S, Pattanaik A, Rehbein J, Reiser O.   +3 more
europepmc   +1 more source

Malononitriles and cyanoacetamides containing isoxazoles and isoxazolines

, 2011
Isoxazoles and isoxazolines have been shown in the literature to be an important scaffold for pharmaceuticals and insecticides, as well as a source of synthetic versatility important to many syntheses. As a substitute for other aromatic rings, isoxazoles
Moores, Lee C.
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