Results 91 to 100 of about 1,834 (212)
trans-Hydroxylation of cyclopent-5-ene[d]isoxazolines [PDF]
The title reaction has been studied as a variant of the cyclopentane ring functionalization of cyclopent-5-ene[d]isoxazolines as the key intermediates in total synthesis of azaand oxo prostaglandin analogues by nitrileoxides approach.
Antonevich, I. P., Nesterova, S. V.
core
Herein, we describe a new strategy to prepare chalcogen-functionalized isoxazolines. The strategy involves the reaction of β,γ-unsaturated oximes with electrophilic selenium and tellurium species, affording 19 new selenium- and tellurium-containing ...
Mikaela Pinz (7429352) +11 more
core +1 more source
Optimising systemic insecticide use to improve malaria control
BackgroundLong-lasting insecticidal nets and indoor residual sprays have significantly reduced the burden of malaria. However, several hurdles remain before elimination can be achieved: mosquito vectors have developed resistance to public health ...
Hannah R Meredith +2 more
doaj +1 more source
The asymmetric synthesis of β-hydroxynitriles remains a challenge in organic synthesis. Herein we report a convenient synthesis of β-hydroxynitriles from enantiomerically enriched 3-unsubstituted 2-isoxazolines via a base-catalyzed ring-opening reaction ...
Antti Pohjakallio (2262703) +2 more
core +1 more source
A novel and efficient Cu(OAc)2-catalyzed oxyazidation of unactivated alkenes was developed. The reactions are easy to conduct, occur under mild conditions, and form azido-substituted isoxazolines in good ...
Liping Zhu (25704) +5 more
core +1 more source
A novel and efficient Cu(OAc)2-catalyzed oxyazidation of unactivated alkenes was developed. The reactions are easy to conduct, occur under mild conditions, and form azido-substituted isoxazolines in good ...
Zhu, Liping +11 more
core +1 more source
Anionic Domino C-O-Heterocyclization Approach for the Synthesis of 5-Vinyl Isoxazolines
5-Vinyl isoxazolines were isolated in high yields through domino nucleophilic addition–anionic C–O-heterocyclization, when allyl organometallics derived from trans-1,4-dihalobutene were reacted with nitrile ...
Kumar, H. +7 more
core +1 more source
Synthesis and Antimicrobial Studies of Some Novel Pyrazoline and Isoxazoline Derivatives
A new series of 1H-3-(4’-substituted phenyl)-5-(6’’-methoxy napthaline)-2-pyrazolines (4a-e) and 1H-3-(4’-substituted phenyl)-5-(6’’-methoxynapthaline)-2-isoxazolines (5a-e) were synthesized by reacting 1-(4’-substituted phenyl)-3-(6’’-methoxynapthaline)-
S. B. jadhav +3 more
doaj +1 more source
3-Fluoro arylcycloopent-5-en[d]isoxazolines have been obtained via the 1,3-dipolar cycloaddition of cyclopentadiene to aromatic nitrile oxides. The reductive cleavage of these isoxazolines by Raney nickel in trifluoroacetic acid led to corresponding ...
Antonevich, I. P. +2 more
core
A One-Pot Approach to Δ2‑Isoxazolines from Ketones and Arylacetylenes
The sequential reaction of ketones with arylacetylenes and hydroxylamine in the presence of KOBut/DMSO followed by the treatment of the reaction mixture with H2O and KOH leads to Δ2-isoxazolines in up to 88 ...
Elena Yu. Schmidt (2007184) +5 more
core +1 more source

