Синтез (2-фторфенил)-и (4-фторфенил)-(2-нитрометилциклопентил)метанонов как предшественников фторсодержащих простаноидов [PDF]
, 2014 Осуществлен синтез новых фторсодержащих первичных нитросоединений ? (2-фторфенил) и (4-фторфенил)-(2-нитрометилциклопентил)метанонов посредством 1,4-присоединения нитрометана к 1-ацилциклопентенам, полученным в результате восстановительного расщепления ...
Антоневич, Инесса Петровна +2 more
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Deep Eutectic Solvents: The Organic Reaction Medium of the Century [PDF]
, 2016 This microreview summarizes the use of deep eutectic solvents (DESs) and related melts in organic synthesis. Solvents of this type combine the great advantages of other proposed environmentally benign alternative solvents, such as low toxicity, high ...
Abbott +192 more
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Syntheses of Isoxazoline-Based Amino Acids by Cycloaddition of Nitrile Oxides and Their Conversion into Highly Functionalized Bioactive Amino Acid Derivatives [PDF]
, 2012 The present account illustrates the syntheses of isoxazoline- based amino acids by the cycloaddition of 1,3-dipolar nitrile oxides to the C–C double bond of unsaturated amino acid derivatives, with focus on the regio- and stereoselectivities of the ...
Fülöp, Ferenc +2 more
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One-step synthesis of differently bis-functionalized isoxazoles by cycloaddition of carbamoylnitrile oxide with β-keto esters [PDF]
, 2012 A new protocol for synthesizing different functionalized isoxazoles is provided. Carbamoylnitrile oxide generated from nitroisoxazolone underwent inverse electron-demand 1,3-dipolar cycloaddition with 1,3-dicarbonyl compounds in the presence of magnesium
975 +15 more
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Aryl nitrile oxide cycloaddition reactions in the presence of pinacol boronic acid ester
Beilstein Journal of Organic Chemistry, 2012 An aryl substrate with dual functionality consisting of a nitrile oxide and a pinacolyl boronate ester was prepared by mild hypervalent iodine oxidation (diacetoxyiodobenzene) of the corresponding aldoxime, without decomposition of the boronate ...
Sarah L. Harding +2 more
doaj +1 more source
Optimising systemic insecticide use to improve malaria control
BMJ Global Health, 2019 BackgroundLong-lasting insecticidal nets and indoor residual sprays have significantly reduced the burden of malaria. However, several hurdles remain before elimination can be achieved: mosquito vectors have developed resistance to public health ...
Hannah R Meredith +2 more
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مجلة بغداد للعلوم, 2016 In this paper some chalcones (C1-C8) are prepared based on the reaction of one mole of substituted acetophenone with one mole of substituted benzaldehydes in the presence of (40%) sodium hydroxide as a base.
Baghdad Science Journal
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Транс-гидроксилирование ряда циклопен-5ЕН[d]изоксазолинов [PDF]
, 2013 Титульная реакция была изучена как вариант функционализации циклопентанового кольца циклопент-5-ен[d]изоксазолинов ? ключевых интермедиатов в полном синтезе азоти кислородсодержащих простаноидов в рамках нитрилоксидного подхода.
Антоневич, Инесса Петровна +1 more
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Sintesis Pirazolin dari Kalkon 3-kloro Inti Naftalen dan Uji Aktivitasnya sebagai Antibakteri [PDF]
, 2014 Pyrazolines have been reported to possess many of interesting biological activities such as antimicrobial, antidepressant, antitumor, antioxidant, antiinflammatory, anticancer and anticonvulsant activity .
Jasril, J. (Jasril) +2 more
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Synthesis of (2-fluorophenyl) and (4-fluorophenyl)-(2-nitromethyl)-methanones as precursors of fluorinated prostanoids [PDF]
, 2014 The synthesis of new fluorinated primary nitrocompounds ?(2-fluorophenyl)and (4-fluorophenyl)-(2-nitromethylcyclopentyl)methanones has been realized by the nitromethane 1,4-addition to 1-acylcyclopentenes, available by the reductive cleavage of ...
Antonevich, I. P. +2 more
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