(7, 8-Dimethyl-2-oxo-2H-chromen-4-yl)methyl morpholine-4-carbodithioate
In the title compound, C17H19NO3S2, the chromene unit makes a dihedral angle of 88.48 (5)° with the best plane through the morpholine ring. The carbodithioate group is present in an antiperiplanar conformation with respect to the morpholine ring, as ...
Shamantha Kumar +4 more
doaj +1 more source
Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones [PDF]
Two series of novel rigid pyrazolone derivatives were synthesized and evaluated as inhibitors of Mycobacterium tuberculosis (MTB), the causative agent of tuberculosis. Two of these compounds showed a high activity against MTB (MIC = 4 μg/mL).
Alessandro De Logu +19 more
core +1 more source
Novel (4-methoxy or 4,8-dimethoxy)-3-methyl-N-(6-oxo-2-thioxo-1,2,3, 6-tetrahydro- pyrimidin-4-yl) benzo [1,2-b: 5, 4-b’] difuran-2-carboxamide (5a−b) has been synthesized by the reaction of visnagenone−ethylacetate (2a) or khellinone ...
Ameen Ali Abu-Hashem +2 more
doaj +1 more source
Application of MEA, TEPA and Morpholine Grafted NaY Zeolite as CO2 Capture [PDF]
In the current research, NaY zeolite with a molar ratio of Si/Al=2.5 was grafted chemically with amines like monoethanolamine, tetraethylenepentamine, and morpholine.The modified NaY zeolites were characterized by XRD, FT-IR, TGA, EDAX, BET, FESEM, CO2 ...
Heshmatollah Alinezhad +3 more
doaj +1 more source
Synthesis and biological evaluation of novel PDMP analogues [PDF]
A new series of hybrid PDMP analogues, based both on PDMP and styryl analogues of natural ceramide, has been synthesized from D-serine. The synthetic route was developed such that future introduction of different aryl groups is straightforward ...
Boldin-Adamsky, Swetlana +5 more
core +1 more source
Dinuclear Lanthanide (III) coordination polymers in a domino reaction [PDF]
A systematic study was performed to further optimise the catalytic room-temperature synthesis of trans-4,5- diaminocyclopent-2-enones from 2-furaldehyde and primary or secondary amines under a non-inert atmosphere. For this purpose, a series of dinuclear
Abdul-Sada, Alaa +5 more
core +2 more sources
2-(4-Isobutylphenyl)-1-(morpholin-4-yl)propan-1-one
In the title compound, C17H25NO2, the morpholine ring adopts a chair conformation. The benzene ring makes a dihedral angle of 39.81 (13)° with the basal plane of the morpholine group.
Nasirullah +4 more
doaj +1 more source
Enterovirus Inhibition by Hinged Aromatic Compounds with Polynuclei
The modern world has no available drugs for the treatment of enteroviruses (EV), which affect millions of people worldwide each year. The EV71 is a major causative disease for hand, foot, and mouth disease; sometimes it is associated with severe central ...
Jih Ru Hwu +8 more
doaj +1 more source
Oxidation of some Alicyclic Amines by Potassium Hexacyanoferrate (III) in Alkaline Medium: A Kinetic and Mechanistic Study [PDF]
Oxidation of some alicyclic amines (morpholine, piperazine and piperidine) by potassium hexacyanoferrate(???) in basic medium has been investigated at 35°C.
M. M. Al-Subu +4 more
doaj +1 more source
Design, synthesis and biological evaluation of 1,3-dihydroxyxanthone derivatives: Effective agents against acetylcholinesterase [PDF]
The present work concerns the rational design and development of new inhibitors of acetylcholinesterase (AChE) based on the privileged xanthone scaffold.
Accordino, Sebastian Roberto +5 more
core +1 more source

