Results 281 to 290 of about 121,181 (303)

IP562083 a novel mGluR7 negative allosteric modulator

Pharmacological Reports, 2015
Piotr Brański, Grzegorz Burnat, Anna Stankiewicz, Ryszard Bugno, Maria Paluchowska, Katarzyna Kaczorowska, Barbara Chruścicka, Andrzej Bojarski, Andrzej Pilc   +8 more
openaire   +1 more source

Small Molecules as Negative Allosteric Modulators of Alpha7 nAChRs

2012
VCU Theses and ...
openaire   +1 more source

Selective mGluR1 Negative Allosteric Modulator Reduces Blood–Brain Barrier Permeability and Cerebral Edema After Experimental Subarachnoid Hemorrhage

Translational Stroke Research, 2019
Cheng Zhang, Ming Jiang, Wei-qi Wang, Shi-jun Zhao, Yan Yin, Qiong-jie Mi, Ming‐feng Yang, Yuqiang Song, Bao-liang Sun, Zong-yong Zhang   +9 more
semanticscholar   +1 more source

Positive and negative allosteric modulation of GluK2 kainate receptors by BPAM344 and antiepileptic perampanel

Cell Reports, 2023
Shanti Pal Gangwar, Maria V Yelshanskaya, Alexander I Sobolevsky   +2 more
exaly  

β-Arrestin-Biased Allosteric Modulator of NTSR1 Selectively Attenuates Addictive Behaviors

Cell, 2020
Lauren M Slosky, Yushi Bai, Krisztián Tóth   +2 more
exaly  

Computer-aided design of negative allosteric modulators of NMDA receptor

Doklady Biochemistry and Biophysics, 2013
E V, Radchenko, D S, Karlov, A N, Zefirov, V A, Palyulin, N S, Zefirov, V M, Pentkovski   +5 more
openaire   +2 more sources

The Negative Allosteric Modulator EU1794-4 Reduces Single-Channel Conductance and Ca2+ Permeability of GluN1/GluN2A N-Methyl-d-Aspartate Receptors

Molecular Pharmacology, 2021
Riley E Perszyk, Miranda J Mcdaniel, Brooke M Katzman   +2 more
exaly  

The GluN1/GluN2B NMDA receptor and metabotropic glutamate receptor 1 negative allosteric modulator has enhanced neuroprotection in a rat subarachnoid hemorrhage model

Experimental Neurology, 2018
Zong-yong Zhang, Junke Liu, Cundong Fan, Leilei Mao, Rong-xia Xie, Suyun Wang, Ming-feng Yang, Hui Yuan, Xiao-yi Yang, Jingyi Sun, Jian Wang, J. Kong, Siluo Huang, Baoliang Sun   +13 more
semanticscholar   +1 more source

Discovery of VU0409106: A negative allosteric modulator of mGlu5 with activity in a mouse model of anxiety

Bioorganic and Medicinal Chemistry Letters, 2013
Andrew S Felts, Ryan D Morrison, Daryl F Venable   +2 more
exaly  

Negative allosteric modulation of the µ-opioid receptor

Biophysical Journal
Evan S. O'Brien, Vipin A. Rangari, Amal El Daibani, Shainnel O. Eans, Betsy White, Haoqing Wang, Yuki Shiimura, Kaavya Krishna Kumar, Kevin Appourchaux, Chensong Zhang, Jesper M. Mathiesen, Tao Che, Jay P. McLaughlin, Susruta Majumdar, Brian K. Kobilka   +14 more
openaire   +1 more source