Results 51 to 60 of about 1,089 (139)
Efficient Synthesis of B-Alkylated Oxazaborolidines Derived from Ephedrine and Norephedrine
Representative B-butyl- and B-methyl-1,3,2-oxazaborolidines derived from ephedrine and norephedrine were prepared in good yield and excellent purity by one-pot treatment of B-H oxazaborolidines with the corresponding organolithium reagent and subsequent ...
Ruth Figueroa (1887805) +6 more
core +1 more source
Helix−Helix Transition of Optically Active Poly((1R,2S)-N-(4-ethynylbenzyl)norephedrine) Induced by Diastereomeric Acid−Base Complexation Using Chiral ...
Yoshio Okamoto (1887238) +2 more
core +2 more sources
ABSTRACT Survivors and refugees of war often have mental, behavioral, emotional, and spiritual consequences from undergoing civil unrest. In many cases, counselors utilize cognitively‐based therapies as the recommended treatment to alleviate these issues.
Isaac Burt, Luis A. Tosado II
wiley +1 more source
Radical-mediated cyclization of norephedrine derived o-bromobenzamide 5 was found to be fairly stereoselective (85:15)favouring diastereoisomer trans-6.
Laura Belvisi +9 more
core +1 more source
Fused nitrogen‐bridgehead N,O‐acetals receive specific emphasis as pivotal scaffolds due to their significant role in the bioactivity of medicinally relevant molecules. Significant approaches have been reported on their role as key synthetic building blocks/motifs in the construction of complex organic molecules and their utility as chiral auxiliaries ...
Alexis D. Kouvelas +2 more
wiley +1 more source
ABSTRACT The synthesis of enantiopure α‐hydroxy ketones, particularly R‐ and S‐phenylacetylcarbinol (PAC), represents an important process in the pharmaceutical industry, serving as a pivotal step in the production of drugs. Recently, two novel enzymes, ephedrine dehydrogenase (EDH) and pseudoephedrine dehydrogenase (PseDH), have been described.
Reynaldo Jr. Carubio +2 more
wiley +1 more source
Radical-mediated cyclization of norephedrine derived alpha-iodoamides 1 was found to be highly stereoselective (> 97.3) favouring diastereoisomer 2. Bicyclic lactams 2 were transformed in high yields into enantiomerically pure pyrrolidines 10. Transition
Laura Belvisi +11 more
core +1 more source
Two‐Step Biocatalytic Synthesis of (1S)‐Nor(pseudo)ephedrine Catalyzed by Immobilized Enzymes
A biocatalytic cascade was designed for the synthesis of (1S,2S)‐norpseudoephedrine [(1S,2S)‐NPE] and (1S,2R)‐norephedrine [(1S,2R)‐NE], involving a benzoin‐type condensation catalyzed by (S)‐selective acetoin:dichlorophenolindophenol oxidoreductase (Ao : DCPIP OR), followed by a transamination mediated by (S)‐ or (R)‐selective amine transaminase (ATA).
Stefania Patti +7 more
wiley +1 more source
The treatment of esters of amino acids with dimethoxytetrahydrofuran furnished pyrrole derivatives of amino acid esters. The Wilsmeier-Haack formylation followed by the reaction of the formylated pyrroles with norephedrine afforded a selective formation ...
N. Tuna Subasi +6 more
core +1 more source
Golden Guardians: Advanced pH Sensors with Built‐in Antimicrobial Defense
Ultrasmall norephedrine‐capped gold nanoclusters (Au@Nore) exhibit high photoluminescence (ΦPL of up to 33%) reversible ratiometric pH sensing and pH‐dependent antimicrobial activity. They enabled us to evaluate the pH sensing and their biological effect on bacteria and yeast. Abstract Gold nanoclusters (Au NCs) capped with a small biomolecule, namely (
Miguel Justo‐Tirado +6 more
wiley +1 more source

