Results 171 to 180 of about 19,199 (236)

Potent <i>in vitro</i> synergistic antiviral effects of the pan-coronavirus fusion inhibitor EK1 in combination with RBD-specific antibodies or M^pro inhibitors. [PDF]

J Virol
Xiu R, Wang Y, Cai W, Wang Q, Xie M, Wang Y, Li C, Wang Q, Huang J, Ying T, Song C, Lu L, Jiang S, Xu W.   +13 more
europepmc   +1 more source

Constrained TACC3 peptidomimetics for a non-canonical protein-protein interface elucidate allosteric communication in Aurora-A kinase. [PDF]

Chem Sci
Gimenez D, Walko M, Miles JA, Bayliss R, Wright MH, Wilson AJ.   +5 more
europepmc   +1 more source

Disrupting the ASH2L-DPY30 PPI in cancer: structure, function, and therapeutic opportunities in H3K4 methylation. [PDF]

Epigenetics Chromatin
Kamel EM, Allam AA, Rudayni HA, Alkhedhairi S, Ahmed NA, Alkhayl FFA, Lamsabhi AM.   +6 more
europepmc   +1 more source

Intermolecular Stacking-Instructed Chiral Preference in Covalent 2 + 2 Macrocyclization. [PDF]

JACS Au
Huang ZS, Wang WR, Yang FH, Gou F, Jiang L, Qiu CC, Tai YY, Yan XS, Wu X, Jiang T, Jiang YB.   +10 more
europepmc   +1 more source

Discovery of highly potent α-keto ester-based peptidomimetic inhibitors of the Hip1 protease for the treatment of <i>Mycobacterium tuberculosis</i>. [PDF]

Eur J Med Chem Rep
Schumann N, Shamma F, Brooks CL, Johnson SJ, Yim MK, Olsen KJ, Peña K, Karakousis PC, Abell A, Goldfarb NE.   +9 more
europepmc   +1 more source

Cell-Mediated and Peptide-Based Delivery Systems: Emerging Frontiers in Targeted Therapeutics. [PDF]

Pharmaceutics
Erdei E, Deme R, Balogh B, Mándity IM.
europepmc   +1 more source

Recognition of the CREB-Binding Protein/Mixed Lineage Leukemia Interface by Sulfonyl-γ-AApeptides: Beyond Mimicry of Mixed Lineage Leukemia. [PDF]

J Med Chem
Huang B, Wang M, Gregory-Lott E, Li BX, Win YY, Shen N, Chen J, Li S, Cao C, Xiao X, Daughdrill GW, Cai J.   +11 more
europepmc   +1 more source

Development of ketobenzothiazole-based peptidomimetic TMPRSS13 inhibitors with low nanomolar potency. [PDF]

J Enzyme Inhib Med Chem
Joushomme A, Désilets A, Champagne W, Hassanzadeh M, Lemieux G, Gravel-Trudeau A, Lepage M, Lafrenière S, Froehlich U, List K, Boudreault PL, Leduc R.   +11 more
europepmc   +1 more source

Opioid Affinity of Diazacyclic Peptidomimetic Compounds Derived from Reduced Polyamides. [PDF]

Int J Mol Sci
Chaudhari P, Bunnell A, Yegambaram M, Dooley C, Nefzi A.   +4 more
europepmc   +1 more source

Fluorine Chemistry. [PDF]

ACS Org Inorg Au
Poisson T, Dichiarante V.
europepmc   +1 more source