Results 171 to 180 of about 12,487 (241)

Advancements in development of novel class of HIV protease inhibitors. [PDF]

Ann Med
Gu WG, Yin GZ, Zhang YP.
europepmc   +1 more source

Native MS and ligand observed NMR uncovers subtle SLiM binding variations that mediate HSP90-Hop PPI modulation. [PDF]

RSC Chem Biol
Davids TK, Kusza DA, Misplon SK, Späth JC, Mhlanga R, Clarke DJ, de la Torre BG, Albericio F, Edkins AL, Rylands M, Veale CGL.   +10 more
europepmc   +1 more source

Fat or flat? The impact of dipole moment vectors on non-covalent interactions between aromatic tags and macromolecules.

Inorg Chem Front
Holub J, Jílková A, Lemke C, Cianni L, Spiwoková P, Horn M, Breuer C, Leontovyč A, Brynda J, Mertlíková-Kaiserová H, Chanová M, Dos Reis Rocho F, Montanari CA, El-Sakkary N, Caffrey CR, Gütschow M, Hnyk D, Mareš M, Fanfrlík J.   +18 more
europepmc   +1 more source

Thiazole peptidomimetics as chemical modulators of <i>KRAS</i> gene expression <i>via</i> G-quadruplex stabilization. [PDF]

RSC Chem Biol
Biswas D, Gorai A, Maiti S, Chaudhuri R, Pradhan S, Dash J.   +5 more
europepmc   +1 more source

Antimicrobial activity of a short guanidine mimic immobilised on contact lenses. [PDF]

J Mater Sci Mater Med
Sara M, Kuppusamy R, Enninful G, Suresh D, Vasilev K, Mackenzie D, Dehghani F, Hui A, Wong EHH, Yasir M, Kumar N, Willcox M.   +11 more
europepmc   +1 more source

Conformational free energy landscape of sorting signal peptides in complex with bacterial sortases. [PDF]

Biophys J
Croney KA, Huisman C, Brock R, Whitham KM, Amacher JF, McCarty J.   +5 more
europepmc   +1 more source

Development of Peptidomimetic PROTACs as Potential Degraders of 3-Chymotrypsin-like Protease of SARS-CoV-2. [PDF]

Int J Mol Sci
Wei C, Li Y, Guo L, Shao Z, Diao H.
europepmc   +1 more source

Integrated computational screen and validation of thalidomide-based PROTACs targeting SARS-CoV-2 main protease. [PDF]

RSC Med Chem
Guo LN, Li YH, Zhu RY, Su N, Shao ZY, Diao H.   +5 more
europepmc   +1 more source

AlphaFold-Guided Discovery of an Overlapping MYC/Miz-1 Interface Enables Peptidomimetic Disruption of MYC/MAX. [PDF]

ChemMedChem
Ellenbroek BD, Tirtosentono ASS, Pomplun SJ.   +2 more
europepmc   +1 more source

Design, Synthesis, and Biological Evaluation of Peptidomimetic Tetrahydropyrrole Spirodihydroindolones as SARS-CoV-2 3CL Protease Inhibitors. [PDF]

ACS Med Chem Lett
Hu L, Zhao Z, Zhang S, Yang L, Cui W, Hu T, Suo J, Sun H, Zhang Q, Zhang L, Zhu W, Xu Z, Zhang Y, Jiang X, Zhang Y, Shen J.   +15 more
europepmc   +1 more source