Indole Peptidomimetics Show Potent and Selective Activity against Drug-Resistant <i>Plasmodium falciparum</i>. [PDF]
Januário MAP +8 more
europepmc +1 more source
Evidence of an activity-enhancing conformational shift in Arabidopsis thaliana plant cysteine oxidase 4 induced by binding of substrate or substrate-mimics. [PDF]
Latter R +8 more
europepmc +1 more source
Biological evaluation of ferrocene peptidomimetics
Peptidomimetici su spojevi čiji esencijalni farmakoforni elementi oponašaju 3D strukturu prirodnog peptida i/ili proteina te zadržavaju njegovu sposobnost interakcije s biološkim ciljanim sustavima, pri čemu zadržavaju jednak ili unaprijeđen biološki ...
Mihalj, Nika
core
Covalent Peptide-Based N-Myc/Aurora-A Inhibitors Bearing Sulfonyl Fluoride Warheads. [PDF]
Dawber RS +6 more
europepmc +1 more source
Covalent Radiopharmaceuticals: Precision Imaging and Therapy for Cancer. [PDF]
Klauser PC, Wang L.
europepmc +1 more source
Using generative AI to transform peptide hits into small molecule leads. [PDF]
Mills J, Lau YH.
europepmc +1 more source
Antimicrobial activity of a short guanidine mimic immobilised on contact lenses. [PDF]
Sara M +11 more
europepmc +1 more source
GPepT: A Foundation Language Model for Peptidomimetics Incorporating Noncanonical Amino Acids. [PDF]
Oikawa Y +8 more
europepmc +1 more source
Antimicrobial nanocoatings and films for contact lenses: progress and promise. [PDF]
Sara M, Attard S, Kumar N, Willcox M.
europepmc +1 more source

