Results 151 to 160 of about 10,137 (233)

Deconvolution of the On-Target Activity of Plasmepsin V Peptidomimetics in <i>Plasmodium falciparum</i> Parasites. [PDF]

ACS Infect Dis
Su W, Nguyen W, Siddiqui G, Dziekan JM, Marapana D, Penington JS, Mehra S, Razook Z, McCann K, Ngo A, Jarman KE, Barry AE, Papenfuss AT, Gilson PR, Creek DJ, Cowman AF, Sleebs BE, Dans MG.   +17 more
europepmc   +1 more source

Bridging Heterocycle-Mediated Hydrogen Bonding Facilitates Permeability of Polar Macrobicycles. [PDF]

J Am Chem Soc
Cooper GID, Dai B, Durham N, Walker GL, Yu H, Mendoza A, Bernardino SJ, Wu YD, Harran PG.   +8 more
europepmc   +1 more source

Opioid Affinity of Diazacyclic Peptidomimetic Compounds Derived from Reduced Polyamides. [PDF]

Int J Mol Sci
Chaudhari P, Bunnell A, Yegambaram M, Dooley C, Nefzi A.   +4 more
europepmc   +1 more source

Blood-Brain Barrier Penetration of Novel 4-Trifluoromethyl-Coumarin Hybrids with Antibacterial Properties as Potential Brain Therapeutics in the Context of Spatially Diverse Healthcare Systems. [PDF]

Int J Mol Sci
Kowalczyk P, Koszelewski D, Misztal T, Szlis M, Młotkowska P, Gołębiewski M, Głowacz K, Kocot M, Marczyk M, Wypych A, Kurylczyk A, Krajewska-Pędzik A, Ostaszewski R.   +12 more
europepmc   +1 more source

Forces behind N- and C-capping of peptidic helices. [PDF]

Chem Commun (Camb)
Mi T, Mattes L, Pewklang T, Hauser K, Burgess K.   +4 more
europepmc   +1 more source

A molecular perspective of gelsolin amyloidosis: An old foe with new faces. [PDF]

Cell Mol Life Sci
Bollati M, Natale C, Girois L, Conz A, Peqini K, Pieraccini S, Pellegrino S, Diomede L, de Rosa M.   +8 more
europepmc   +1 more source

SOCS1-based therapeutic peptides improve liver disease and metabolic dysfunction in obesity and diabetes. [PDF]

Sci Rep
Soto-Catalán M, Opazo-Ríos L, Espadas C, Romero-Cote M, Lázaro I, Moreno JA, Gómez-Guerrero C, Egido J, Mas-Fontao S.   +8 more
europepmc   +1 more source

Role of Structural Modifications in Peptidomimetic Compounds as Potential Antimicrobial Agents against <i>Staphylococcus aureus</i> and <i>Streptococcus pyogenes</i>: Balancing Bioavailability, Safety, and Antimicrobial Activity. [PDF]

ACS Omega
Dzierżyńska M, Sawicka J, Łada K, Gajewicz-Skretna A, Deptuła M, Chernobrovkin A, Pogorzelska A, Grubb A, Zubarev RA, Pikuła M, Kasprzykowski F, Rodziewicz-Motowidło S.   +11 more
europepmc   +1 more source

Breaking biofilm barriers in skin wounds: Membrane-Active antimicrobials in an era of resistance. [PDF]

Curr Res Pharmacol Drug Discov
Hemmingsen LM, Škalko-Basnet N.
europepmc   +1 more source

Thiazole peptidomimetics as chemical modulators of <i>KRAS</i> gene expression <i>via</i> G-quadruplex stabilization. [PDF]

RSC Chem Biol
Biswas D, Gorai A, Maiti S, Chaudhuri R, Pradhan S, Dash J.   +5 more
europepmc   +1 more source