Results 121 to 130 of about 52,734 (205)

Stereocontrolled entry to borylated piperidines <i>via</i> stepwise dearomative carboboration of pyridines. [PDF]

Chem Sci
Khalse LD, DeSnoo W, Lou YP, Tantillo DJ, Nairoukh Z.   +4 more
europepmc   +1 more source

An orally available PfPKG inhibitor blocks Plasmodium's infection of the liver. [PDF]

PLoS Pathog
Dhiyebi H, Mbaye A, Thaniana A, Gilleran J, Eck T, Ashraf K, Kudyba K, Fan H, Seibold S, Battaile KP, Siekierka J, Johnson E, Roth A, De Rocher A, Lovell S, Miller EB, Roberge JY, Bhanot P.   +17 more
europepmc   +1 more source

Structural Modification of Sesquiterpene Lactones via Michael Addition: Improved Bioactivity and Pharmacokinetics. [PDF]

Int J Mol Sci
Ha MW, Kang J, Lee S, Paek SM.
europepmc   +1 more source

Design, Synthesis, and Biological Activity of Isothiocyanate-Triazine Conjugates as AChE and BACE1 Inhibitors. [PDF]

Biomolecules
Górecki K, Polakowski J, Więckowska N, Grzywa R, Frączyk J, Kolesińska B, Wróbel-Tałałaj A, Drozdowska D, Janczewski Ł.   +8 more
europepmc   +1 more source

Direct Access to Chiral Piperidines by Enantioselective HAT-Initiated C(sp³)─H Oxidation. [PDF]

Angew Chem Int Ed Engl
Muthuramalingam S, Luis JM, Call A, Lefebvre Q, Sigman MS, Costas M.   +5 more
europepmc   +1 more source

Decoding Prolonged Residence Time of 5-HT_2A Receptor Antagonists: Insights from Ritanserin Derivatives. [PDF]

J Chem Inf Model
Kordylewski SK, Kurowska K, Nędza K, Satała D, Bugno R, Podlewska S.   +5 more
europepmc   +1 more source

Synthesis and Evaluation of Novel Cinnamic Acid Hybrids With Antiacetylcholinesterase, Antioxidant, and Anti-Inflammatory Properties. [PDF]

ChemMedChem
Sdougkou K, Rekka E, Papagiannopoulou D.
europepmc   +1 more source

Toward Chromatography-Free Convergent Peptide Synthesis via Nanostar Sieving. [PDF]

Org Process Res Dev
Al-Kadhimi M, Botwright J, Oxley A, Ju Han S, Tandogan Gray N, Frederick MO, Peeva L, Livingston AG.   +7 more
europepmc   +1 more source

Novel 3‑Heteroaryl Pyrrolidine and Piperidine Compounds as Orexin Receptor Agonists for Treating Sleep Disorders, namely, Narcolepsy and Hypersomnia. [PDF]

ACS Med Chem Lett
Sabnis RW.
europepmc   +1 more source

Deaminative Fluorination of Sulfonamides via Aminocyclopropenium Activation. [PDF]

Org Lett
Carneiro SN, Bento JV, Zimmerman PM, Sanford MS.   +3 more
europepmc   +1 more source