Results 1 to 10 of about 1,984 (207)
Synthesis and Adrenolytic Activity of New Propanolamines [PDF]
Molecules, 2010 The synthesis of (2R,S)-1-(6-methoxy-4-(methoxymethyl)-1H-indol-5-yloxy)-3-(2-(2-methoxyphenoxy)ethylamino)propan-2-ol and (2R,S)-1-(4-methoxy-6-(methoxymethyl)-1H-indol-5-yloxy)-3-(2-(2-methoxyphenoxy)ethylamino)propan-2-ol is described.
Grażyna Groszek +6 more
doaj +7 more sources
Enantiomeric Propanolamines as selectiveN-Methyl-
Journal of Medicinal Chemistry, 2008 Enantiomeric propanolamines have been identified as a new class of NR2B-selective NMDA receptor antagonists. The most effective agents are biaryl structures, synthesized in six steps with overall yields ranging from 11-64%. The compounds are potent and selective inhibitors of NR2B-containing recombinant NMDA receptors with IC 50 values between 30-100 ...
Yesim A. Tahirovic +17 more
semanticscholar +5 more sources
ANTIMICROBIAL PROPERTIES OF BUTANOLAMINES AND PROPANOLAMINES IN METAL WORKING FLUIDS
The Journal of General and Applied Microbiology, 1979 Seventeen propanolamines, six diisopropanolamines, and two butanolamines were studied for their antimicrobial properties against a mixed flora of fungi and bacteria in cutting fluids. All of the propanolamines showed inhibitory properties in the lubricants.
E. O. Bennett, M.C. Adams, G. Tavana
semanticscholar +5 more sources
SOME PHARMACOLOGICAL PROPERTIES OF 3:3‐DIPHENYL‐PROPANOLAMINES, ‐ALLYLAMINES, AND ‐PROPYLAMINES [PDF]
British Journal of Pharmacology and Chemotherapy, 1951 This programme was undertaken with the knowledge that some compounds containing this structure exhibit pharmacological activity. This is exemplified by Hochst 10116 (Ph2CH.CH2CH2NCH2), which is a component of the anti-asthmatic mixture "Aspasan," in ...
A. C. White, A. F. GREEN, A.G. Hudson
semanticscholar +6 more sources
Synthesis and adrenergic .BETA.-blocking activity of some propanolamine derivatives.
Chemical and Pharmaceutical Bulletin, 1978 Some propanolamine derivatives were synthesized and their β-adrenergic blocking activities were determined. Among the compounds tested, all compounds with benzothiazole nucleus were found to have potent β-adrenergic blocking activity, and those with other nuclei failed to produce substantial β-blocking activity with one exception.
H. OBASE +7 more
openalex +5 more sources
RSC Advances, 2020 Various 1,4-benzoxazin-3-one derivatives containing propanolamine groups have been shown to exhibit good antibacterial activity againstPseudomonas syringaepvactinidiae(Psa),X. axonopodispvcitri(Xac) andXanthomonas oryzaepvoryzae(Xoo).
Jia‐Rui Rao +5 more
openalex +5 more sources
Journal of Cardiovascular Pharmacology, 2002 A propanolamine derivative with vanillylamide base, KMUP 880602, was first investigated under in vivo and in vitro conditions. IV KMUP 880602 (0.1, 0.5, 1.0, and 2.0 mg/kg) produced dose-dependent hypotensive and bradycardia responses in pentobarbital-anesthetized Wistar rats. KMUP 880602 also markedly inhibited both the tachycardia effects induced by (
Jwu‐Lai Yeh +7 more
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(11)Preparation of Propanolamine Oleate
The Journal of the Society of Chemical Industry, Japan, 1952 Masumi Saito, Minoru Imoto
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Studies of some beta-propanolamines, imidazo [2,1-b] thiazoles and ylides, by X-ray analysis [PDF]
, 1975 In this thesis, single crystal X-ray diffraction techniques have been used to determine the crystal and molecular structures of ten compounds. The contents are presented in four Parts, the first of which is a brief discussion on some theoretical aspects ...
I. R. Cameron
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Densities, Viscosities of Pure 1-(2-Hydroxyethyl) Pyrrolidine, 3-Amino-1-Propanol, Water, and Their Mixtures at 293.15 to 363.15 K and Atmospheric Pressure [PDF]
, 2023 Densities and viscosities of pure 1-(2-hydroxyethyl) pyrrolidine, 3-amino-1-propanol, water, and their blends’ data are reported from 293.15 to 363.15 K and at ambient pressure.
Hartono, Ardi, Knuutila, Hanna K
core +1 more source