Results 1 to 10 of about 1,956 (206)
Synthesis and Adrenolytic Activity of New Propanolamines [PDF]
Molecules, 2010 The synthesis of (2R,S)-1-(6-methoxy-4-(methoxymethyl)-1H-indol-5-yloxy)-3-(2-(2-methoxyphenoxy)ethylamino)propan-2-ol and (2R,S)-1-(4-methoxy-6-(methoxymethyl)-1H-indol-5-yloxy)-3-(2-(2-methoxyphenoxy)ethylamino)propan-2-ol is described.
Grażyna Groszek +6 more
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Enantiomeric Propanolamines as selectiveN-Methyl-
Journal of Medicinal Chemistry, 2008 Enantiomeric propanolamines have been identified as a new class of NR2B-selective NMDA receptor antagonists. The most effective agents are biaryl structures, synthesized in six steps with overall yields ranging from 11-64%.
Yesim A. Tahirovic +17 more
semanticscholar +5 more sources
SOME PHARMACOLOGICAL PROPERTIES OF 3:3‐DIPHENYL‐PROPANOLAMINES, ‐ALLYLAMINES, AND ‐PROPYLAMINES [PDF]
British Journal of Pharmacology and Chemotherapy, 1951 This programme was undertaken with the knowledge that some compounds containing this structure exhibit pharmacological activity. This is exemplified by Hochst 10116 (Ph2CH.CH2CH2NCH2), which is a component of the anti-asthmatic mixture "Aspasan," in ...
A. C. White, A. F. GREEN, A.G. Hudson
semanticscholar +6 more sources
ANTIMICROBIAL PROPERTIES OF BUTANOLAMINES AND PROPANOLAMINES IN METAL WORKING FLUIDS
The Journal of General and Applied Microbiology, 1979 Seventeen propanolamines, six diisopropanolamines, and two butanolamines were studied for their antimicrobial properties against a mixed flora of fungi and bacteria in cutting fluids.
E. O. Bennett, M.C. Adams, G. Tavana
semanticscholar +5 more sources
Synthesis and adrenergic .BETA.-blocking activity of some propanolamine derivatives.
Chemical and Pharmaceutical Bulletin, 1978 Some propanolamine derivatives were synthesized and their β-adrenergic blocking activities were determined. Among the compounds tested, all compounds with benzothiazole nucleus were found to have potent β-adrenergic blocking activity, and those with other nuclei failed to produce substantial β-blocking activity with one exception.
H. OBASE +7 more
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CATECHOL‐SUBSTITUTED PHENOXY‐PROPANOLAMINES: ADRENOCEPTOR ACTIVITY IN THE ANAESTHETIZED CAT [PDF]
British Journal of Pharmacology, 1977 1 The pharmacological actions of racemic noradrenaline, adrenaline, isoprenaline and N‐t‐butylnoradrenaline have been compared with those of their corresponding derivatives containing an oxymethylene (OXY) link between the ring and ethanolamine side ...
H. Dowd, G. S. Keh, C. Raper
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RSC Advances, 2020 Various 1,4-benzoxazin-3-one derivatives containing propanolamine groups have been shown to exhibit good antibacterial activity againstPseudomonas syringaepvactinidiae(Psa),X. axonopodispvcitri(Xac) andXanthomonas oryzaepvoryzae(Xoo).
Jia‐Rui Rao +5 more
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Journal of Cardiovascular Pharmacology, 2002 A propanolamine derivative with vanillylamide base, KMUP 880602, was first investigated under in vivo and in vitro conditions. IV KMUP 880602 (0.1, 0.5, 1.0, and 2.0 mg/kg) produced dose-dependent hypotensive and bradycardia responses in pentobarbital-anesthetized Wistar rats. KMUP 880602 also markedly inhibited both the tachycardia effects induced by (
Jwu‐Lai Yeh +7 more
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Aryl propanolamines: comparison of activity at human β3 receptors, rat β3 receptors and rat atrial receptors mediating tachycardia [PDF]
British Journal of Pharmacology, 1999 Marlene L. Cohen +4 more
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(11)Preparation of Propanolamine Oleate
The Journal of the Society of Chemical Industry, Japan, 1952 Masumi Saito, Minoru Imoto
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